SCHEMBL20839724

SCHEMBL20839724

CCOC(=O)CCc1cccc(NC(=O)c2ccccc2NC(=O)c2cnc3ccccc3c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.52
CYP2C8 P10632 2/20 0.52
CYP2C19 P33261 2/20 0.52
CYP2C9 P11712 1/20 0.52
NR1H4 Q96RI1 7/20 0.51
PPARG P37231 4/20 0.51
PPARA Q07869 4/20 0.51
ABCB1 P08183 5/20 0.51
ABCG2 Q9UNQ0 4/20 0.51
PPARD Q03181 6/20 0.49
BRAF P15056 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839492 0.87 NR1H4 (0.64) CYP3A4CYP2C8CYP2C19CYP2C9NR1H4
SCHEMBL20839988 0.81 NR1H4 (0.67) NR1H4PPARGPPARAPPARD
SCHEMBL20839936 0.79 NR1H4 (0.65) NR1H4PPARGPPARAPPARD
SCHEMBL20839675 0.79 NR1H4 (0.81) NR1H4PPARGPPARAABCG2PPARD
SCHEMBL20840618 0.79 NR1H4 (0.59) NR1H4PPARGPPARAPPARD
SCHEMBL20839596 0.78 NR1H4 (0.57) NR1H4PPARGPPARAABCG2PPARD
SCHEMBL20839618 0.78 NR1H4 (0.53) NR1H4PPARGPPARAABCG2PPARD
SCHEMBL20839731 0.78 NR1H4 (0.80) NR1H4PPARGPPARAPPARD
SCHEMBL20839717 0.78 NR1H4 (0.70) NR1H4PPARGPPARAABCG2PPARD
SCHEMBL20839943 0.75 FADS1 (0.52) NR1H4PPARGPPARAABCG2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed