SCHEMBL2084795

SCHEMBL2084795

Cc1cc(Cl)cnc1CC(NCCCCN(C)C(=O)OC(C)(C)C)c1nccc2ccccc12

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.33
S1PR3 Q99500 1/20 0.32
AURKA O14965 3/20 0.31
RPS6KB1 P23443 3/20 0.31
ADORA3 P0DMS8 1/20 0.31
TRPV4 Q9HBA0 1/20 0.31
SSTR3 P32745 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
POLB P06746 1/20 0.30
RAD52 P43351 1/20 0.30
KMT2A Q03164 1/20 0.30
UHRF1 Q96T88 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2085959 0.92 GBA1 (0.34) GBA1AURKARPS6KB1ADORA3TRPV4
SCHEMBL2085673 0.80 CXCR4 (0.33) NPC1RAB9APOLBRAD52KMT2A
SCHEMBL2084797 0.80 CXCR4 (0.36) GBA1S1PR3AURKARPS6KB1ADORA3
SCHEMBL2084498 0.75
SCHEMBL2084235 0.75 BCHE (0.34) S1PR3TRPV4KMT2A
SCHEMBL2085960 0.72 CXCR4 (0.38) GBA1ADORA3TRPV4KMT2A
SCHEMBL2084400 0.69 SLC40A1 (0.40) NPC1RAB9AKMT2A
SCHEMBL2086441 0.68 CXCR4 (0.36) POLBRAD52KMT2AUHRF1CYP3A4
SCHEMBL2083940 0.68 HCRTR1 (0.36)
SCHEMBL2084362 0.68 BRD4 (0.35) KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-B1 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORP (US) 2021-06-02 EP disclosed
US-7863293-B2 CXCR4 chemokine receptor binding compounds GENZYME CORPORATION (US) 2011-01-04 US disclosed
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
US-20080255197-A1 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED CORPORATION (CA) 2008-10-16 US disclosed
US-7291631-B2 CXCR4 chemokine receptor binding compounds GENZYME CORPORATION (US) 2007-11-06 US disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed
US-20040209921-A1 CXCR4 chemokine receptor binding comounds ANORMED CORPORATION (CA) 2004-10-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209921-A1 CXCR4 chemokine receptor binding comounds CXCR4, CXCR1, CXCR3 GBA1 3802/4885S1PR3 125/4885AURKA 4523/4885
US-20080255197-A1 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS CXCR4, CXCR1, CXCR3 GBA1 2788/4885S1PR3 101/4885AURKA 3929/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.