SCHEMBL20850671

SCHEMBL20850671

C=C(c1ccccc1)c1cn(Cc2ccccc2)c2ccc(Nc3ccc(Cl)cc3C(=O)OC)cc12

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 4/20 0.45
LMNA P02545 3/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
CPT1A P50416 1/20 0.40
ADORA1 P30542 1/20 0.40
P2RX7 Q99572 1/20 0.39
SERPINE1 P05121 1/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15712242 0.91 LMNA (0.52) P2RX3LMNAALDH1A1MAPTCA12
SCHEMBL15712251 0.85 P2RX3 (0.47) P2RX3LMNAALDH1A1MAPTCA12
SCHEMBL15712243 0.82 P2RX3 (0.49) P2RX3LMNAALDH1A1MAPTCA9
SCHEMBL8358799 0.80 NR4A2 (0.53) LMNAALDH1A1MAPTCA12CA1
SCHEMBL15712210 0.79 ERBB2 (0.48) P2RX3LMNAMAPTP2RX7SMN1; SMN2
SCHEMBL15712464 0.77 NR1I2 (0.56)
SCHEMBL15712217 0.77 POLB (0.43) P2RX3LMNAMAPTP2RX7SMN1; SMN2
SCHEMBL15712354 0.76 MAPT (0.49) P2RX3LMNAALDH1A1MAPTP2RX7
SCHEMBL15712637 0.75 ERBB2 (0.50) P2RX3LMNAP2RX7SMN1; SMN2
SCHEMBL15712713 0.75 HDAC1 (0.47) P2RX3LMNAALDH1A1MAPTCA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2915804-B1 NOVEL AMINE DERIVATIVE OR SALT THEREOF AS TNF ALPHA INHIBITORS FUJIFILM TOYAMA CHEMICAL CO LTD (JP) 2019-03-27 EP disclosed