SCHEMBL20855136

SCHEMBL20855136

Cc1ccc(O)cc1-c1ccc2nc(N)sc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.65
GAA P10253 1/20 0.65
L3MBTL1 Q9Y468 1/20 0.65
PIK3CA P42336 11/20 0.62
PIK3CD O00329 10/20 0.62
PIK3CB P42338 9/20 0.62
PIK3CG P48736 8/20 0.62
ABL1 P00519 1/20 0.55
KIT P10721 1/20 0.55
PDGFRA P16234 1/20 0.55
PI4KA P42356 11/20 0.53
PI4KB Q9UBF8 11/20 0.53
MAPT P10636 2/20 0.53
RAB9A P51151 1/20 0.53
PIP5K1C O60331 4/20 0.51
BRD4 O60885 1/20 0.50
APP P05067 1/20 0.49
ALKBH5 Q6P6C2 1/20 0.48
FTO Q9C0B1 1/20 0.48
ALDH1A1 P00352 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20855252 0.82 ABL1 (0.58) HTTGAAL3MBTL1PIK3CAPIK3CD
SCHEMBL3306309 0.81 PIK3CA (0.74) HTTGAAL3MBTL1PIK3CAPIK3CD
SCHEMBL31298 0.80 HTT (1.00) HTTGAAL3MBTL1PIK3CAPIK3CD
Hydrochloric Acid SCHEMBL11729261 0.78 HTT (0.96) HTTGAAL3MBTL1PIK3CAPIK3CD
SCHEMBL20865379 0.78 PIK3CD (0.62) PIK3CAPIK3CDPIK3CBPIK3CGABL1
SCHEMBL20887499 0.77 DYRK1A (0.72) PIK3CAPIK3CGABL1KITPDGFRA
SCHEMBL29646253 0.77 PIK3CA (0.82) HTTGAAL3MBTL1PIK3CAPIK3CD
SCHEMBL5532470 0.77 PIK3CA (0.82) HTTGAAL3MBTL1PIK3CAPIK3CD
SCHEMBL20855175 0.75 CYP3A4 (0.47) HTTGAAPIK3CAPIK3CDPIK3CB
SCHEMBL20855178 0.75 PIK3CA (0.64) HTTGAAPIK3CAPIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111315727-B Benzothiazole compounds and methods of treating neurodegenerative diseases using the same 第一生物治疗股份有限公司 2023-09-29 CN disclosed
EP-3692023-B1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1ST BIOTHERAPEUTICS INC (KR) 2023-05-17 EP disclosed
EP-3692023-B1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1ST BIOTHERAPEUTICS INC (KR) 2023-05-17 EP disclosed
US-10968188-B2 Benzothiazol compounds and methods using the same for treating neurodegenerative disorders 1ST Biotherapeutics, Inc. (KR) 2021-04-06 US disclosed
US-10968188-B2 Benzothiazol compounds and methods using the same for treating neurodegenerative disorders 1ST Biotherapeutics, Inc. (KR) 2021-04-06 US disclosed
US-20200270222-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1ST Biotherapeutics, Inc. 2020-08-27 US disclosed
US-20200270222-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1ST Biotherapeutics, Inc. 2020-08-27 US disclosed
EP-3692023-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1st Biotherapeutics, Inc. (KR) 2020-08-12 EP disclosed
US-10669246-B2 Benzothiazol compounds and methods using the same for treating neurodegenerative disorders 1ST Biotherapeutics, Inc. (KR) 2020-06-02 US disclosed
US-10669246-B2 Benzothiazol compounds and methods using the same for treating neurodegenerative disorders 1ST Biotherapeutics, Inc. (KR) 2020-06-02 US disclosed
WO-2019070093-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1ST Biotherapeutics, Inc. (KR) 2019-04-11 WO disclosed
WO-2019070093-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1ST Biotherapeutics, Inc. (KR) 2019-04-11 WO disclosed
US-20190100500-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1ST Biotherapeutics, Inc. 2019-04-04 US disclosed
US-20190100500-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS 1ST Biotherapeutics, Inc. 2019-04-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190100500-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS ABL2, ABL1, MAPT HTT 20/4885GAA 254/4885L3MBTL1 1651/4885
US-10669246-B2 Benzothiazol compounds and methods using the same for treating neurodegenerative disorders ABL2, ABL1, MAPT HTT 20/4885GAA 254/4885L3MBTL1 1651/4885
US-10968188-B2 Benzothiazol compounds and methods using the same for treating neurodegenerative disorders ABL2, ABL1, MAPT HTT 20/4885GAA 254/4885L3MBTL1 1651/4885
US-20200270222-A1 BENZOTHIAZOL COMPOUNDS AND METHODS USING THE SAME FOR TREATING NEURODEGENERATIVE DISORDERS ABL2, ABL1, MAPT HTT 20/4885GAA 254/4885L3MBTL1 1651/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.