SCHEMBL20855751

SCHEMBL20855751

COc1ccc(Cl)cc1[C@H]1CO1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.43
ALDH1A1 P00352 4/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HTR2B P41595 4/20 0.40
HTR2C P28335 4/20 0.40
PDE1B Q01064 2/20 0.40
PDE2A O00408 1/20 0.40
PDE8B O95263 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CYP2C19 P33261 1/20 0.40
PDE1A P54750 1/20 0.40
PDE4D Q08499 1/20 0.40
PDE1C Q14123 1/20 0.40
PDE11A Q9HCR9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20855753 1.00 TP53 (0.43) TP53ALDH1A1HTR3EHTR3BHTR3A
SCHEMBL30036752 0.80 CYP2C19 (0.52) ALDH1A1MEN1KMT2ACYP2C19KDM4E
SCHEMBL8423985 0.80 CYP2C19 (0.52) ALDH1A1MEN1KMT2ACYP2C19KDM4E
SCHEMBL13651802 0.79 TP53 (0.39) TP53ALDH1A1HTR3EHTR3BHTR3A
SCHEMBL18820312 0.79 SLC6A2 (0.58) HTR2BHTR2CHTR2ASLC6A2SLC6A4
SCHEMBL18908535 0.79 MEN1 (0.48) ALDH1A1MEN1KMT2AKDM4EPOLB
SCHEMBL83692 0.79 MEN1 (0.48) ALDH1A1MEN1KMT2AKDM4EPOLB
SCHEMBL13686388 0.77 ACHE (0.44) ALDH1A1MEN1KMT2AKDM4EPOLB
SCHEMBL12309442 0.75 KDM1A (0.47) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7049820 0.75 TP53 (0.42) TP53ALDH1A1HTR2BHTR2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019063748-A1 ROR-GAMMA INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-04-04 WO disclosed
WO-2019063748-A1 ROR-GAMMA INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-04-04 WO disclosed