SCHEMBL13686388

SCHEMBL13686388

COc1cc(Cl)cc([C@@H]2CO2)c1OC

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.44
PTPN1 P18031 1/20 0.44
PTAFR P25105 2/20 0.42
CYP3A4 P08684 3/20 0.39
MAPK3 P27361 1/20 0.38
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
PTGS2 P35354 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAP3K14 Q99558 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20855753 0.77 TP53 (0.43) ALDH1A1POLBMEN1KMT2AKDM4E
SCHEMBL20855751 0.77 TP53 (0.43) ALDH1A1POLBMEN1KMT2AKDM4E
SCHEMBL1541914 0.74 ACHE (0.59) ACHEPTAFRCYP3A4ALDH1A1PTGS2
SCHEMBL6822928 0.72 PTAFR (0.69) ACHEPTPN1PTAFRCYP3A4MAPK3
SCHEMBL7786361 0.71 CYP19A1 (0.49) ACHEPTPN1MAPK3MAPK1ALDH1A1
SCHEMBL22984885 0.69 HTR2A (0.40) ACHEPTPN1ALDH1A1MEN1KMT2A
SCHEMBL14189350 0.67 ACHE (0.50) ACHECYP3A4ALDH1A1PTGS2MAP3K14
SCHEMBL7779150 0.67 MEN1 (0.35) ACHEPTPN1MAPK3MAPK1ALDH1A1
SCHEMBL25934295 0.66 KDM4E (0.47) ACHECYP3A4MAPK1ALDH1A1PTGS2
SCHEMBL7056856 0.66 ALDH1A1 (0.46) CYP3A4ALDH1A1POLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2103596-A1 Process for the preparation of N-(phenylethyl) anilines salts and solvates thereof useful as serotonin 5-HT6 antagonists Laboratorios Del. Dr. Esteve, S.A. (ES) 2009-09-23 EP disclosed