SCHEMBL20855752

SCHEMBL20855752

COCC(N)c1cc(F)ccc1OC

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GNRHR P30968 1/20 0.40
ADRA2A P08913 2/20 0.38
ADRA1A P35348 2/20 0.38
KDM4E B2RXH2 1/20 0.38
SLC6A2 P23975 4/20 0.38
SLC6A4 P31645 4/20 0.38
SLC6A3 Q01959 3/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 1/20 0.38
CYP2D6 P10635 1/20 0.37
NFE2L2 Q16236 1/20 0.37
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
BLM P54132 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13343117 0.82 KDM4E (0.40) GNRHRADRA2AADRA1AKDM4ESLC6A2
SCHEMBL20855722 0.81 ADRA2A (0.40) GNRHRADRA2AADRA1AKDM4ESLC6A2
SCHEMBL14983853 0.81 SLC6A2 (0.40) GNRHRADRA2AADRA1AKDM4ESLC6A2
SCHEMBL30963569 0.80 CA1 (0.46) SMN1; SMN2
SCHEMBL20855412 0.80 SCN4A (0.42) ADRA2AADRA1AKDM4ECYP2D6MEN1
SCHEMBL20855556 0.80 KDM4E (0.43) SMN1; SMN2ADRA2AADRA1AKDM4ECYP2D6
SCHEMBL20855410 0.80 SCN4A (0.42) ADRA2AADRA1AKDM4ECYP2D6MEN1
SCHEMBL28491946 0.80 PDCD1LG2 (0.39) GNRHRADRA2AADRA1AKDM4ESLC6A2
SCHEMBL28491947 0.80 PDCD1LG2 (0.39) GNRHRADRA2AADRA1AKDM4ESLC6A2
SCHEMBL30152526 0.80 PDCD1LG2 (0.39) GNRHRADRA2AADRA1AKDM4ESLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019063748-A1 ROR-GAMMA INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-04-04 WO disclosed
WO-2019063748-A1 ROR-GAMMA INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-04-04 WO disclosed