SCHEMBL20879769

SCHEMBL20879769

C[C@H](CC#N)c1ccc(C#N)nc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.35
EPHX2 P34913 1/20 0.35
AR P10275 1/20 0.34
PIK3CD O00329 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
HCK P08631 1/20 0.33
SRC P12931 1/20 0.33
KDR P35968 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
MTOR P42345 1/20 0.33
EPHB4 P54760 1/20 0.33
PRKDC P78527 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
PBRM1 Q86U86 1/20 0.33
KDM5B Q9UGL1 1/20 0.32
CHEK1 O14757 4/20 0.32
PGGT1B P53609 1/20 0.32
ATM Q13315 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171647 1.00 KDM4C (0.35) KDM4CEPHX2ARPIK3CDABL1
SCHEMBL20372862 0.84 ALDH1A1 (0.43) EPHX2ARPIK3CDABL1EGFR
SCHEMBL12251238 0.83 EPHX2 (0.34) KDM4CEPHX2ARPIK3CDABL1
SCHEMBL18552809 0.81 EPHX2 (0.37) EPHX2ARPIK3CDABL1EGFR
SCHEMBL20963164 0.80 ESR1 (0.35) EPHX2ARPIK3CDABL1EGFR
SCHEMBL18599607 0.80 ESR1 (0.33) EPHX2ARPIK3CDABL1EGFR
SCHEMBL104694 0.80 PANK3 (0.39) EPHX2ARPIK3CDABL1EGFR
SCHEMBL20879770 0.79 PBRM1 (0.33) EPHX2ARPBRM1CHEK1EGLN2
SCHEMBL18602334 0.79 CHEK1 (0.32) EPHX2ARPIK3CDABL1EGFR
SCHEMBL169697 0.79 SMN1; SMN2 (0.36) ARALDH1A1CYP2D6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3838903-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVE AS JANUS KINASE INHIBITOR Incyte Holdings Corporation (US) 2021-06-23 EP disclosed
EP-3466953-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVE AS JANUS KINASE INHIBITOR Incyte Holdings Corporation (US) 2019-04-10 EP disclosed