SCHEMBL20882004

SCHEMBL20882004

Cc1cc(CCC(=O)NN)ccc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
GAA P10253 1/20 0.51
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
HCAR2 Q8TDS4 1/20 0.47
KDM1A O60341 1/20 0.46
IAPP P10997 3/20 0.45
ALOX5 P09917 1/20 0.44
OR51E2 Q9H255 1/20 0.44
ERCC1 P07992 1/20 0.42
ERCC4 Q92889 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12832384 0.85 ESR1 (0.56) HIF1ACYP1A2ESR1ESR2HCAR2
SCHEMBL23067196 0.85 IAPP (0.57) HIF1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28659512 0.81 ESR1 (0.55) ESR1ESR2HCAR2IAPPALOX5
SCHEMBL755804 0.81 GAA (0.64) HIF1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28055334 0.81 SKP2 (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1358498 0.81 HIF1A (0.52) HIF1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8340607 0.80 GAA (0.71) HIF1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1696094 0.80 ESR1 (0.57) HIF1ACYP1A2CYP3A4ESR1ESR2
SCHEMBL11218783 0.80 THRA (0.57) ESR1ESR2IAPPTHRATHRB
SCHEMBL12246749 0.79 MAPT (0.65) HIF1ACYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068443-B1 RESIDUALIZING LINKERS AND USES THEREOF CENTRE FOR PROBE DEV AND COMMERCIALIZATION (CA) 2019-04-10 EP disclosed