SCHEMBL208852

SCHEMBL208852

O=C1C(c2ccccc2)c2ccccc2N1c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 2/20 0.42
GFER P55789 1/20 0.42
GAA P10253 4/20 0.41
NPSR1 Q6W5P4 2/20 0.41
CES2 O00748 1/20 0.41
BCHE P06276 1/20 0.41
CES1 P23141 1/20 0.41
HPGD P15428 1/20 0.40
MGLL Q99685 1/20 0.39
POLB P06746 2/20 0.39
MAOA P21397 1/20 0.39
ATM Q13315 1/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29915861 1.00 MEN1 (0.44) MEN1KMT2AALDH1A1GFERGAA
SCHEMBL17074881 0.89 MEN1 (0.44) MEN1KMT2AALDH1A1GAANPSR1
SCHEMBL6524996 0.85 CHEK1 (0.41) MEN1KMT2AALDH1A1GFERGAA
SCHEMBL29886595 0.85 CHEK1 (0.41) MEN1KMT2AALDH1A1GFERGAA
SCHEMBL11482347 0.83 KMT2A (0.45) MEN1KMT2AALDH1A1GAANPSR1
SCHEMBL17583721 0.83 ESR1 (0.39) MEN1KMT2AALDH1A1GAANPSR1
SCHEMBL31717971 0.81 MEN1 (0.41) MEN1KMT2AALDH1A1GAANPSR1
SCHEMBL28703009 0.80 ESR1 (0.35) MEN1KMT2AALDH1A1GAANPSR1
Hydrochloric Acid SCHEMBL7503502 0.79 MEN1 (0.44) MEN1KMT2AALDH1A1GAANPSR1
SCHEMBL32677307 0.78 MEN1 (0.47) MEN1KMT2AALDH1A1GFERGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240180894-A1 METHODS OF TREATING MENTAL AND/OR MOOD DISORDERS USING 2-BROMO-LSD ALONE OR IN COMBINATION WITH A MTOR INHIBITOR BETTERLIFE PHARMA INC (CA) 2024-06-06 US disclosed
US-11260027-B2 Donor organ pre-treatment formulation MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2022-03-01 US disclosed
US-11214805-B2 Targeted nanocarriers for the administration of immunosuppressive agents MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2022-01-04 US disclosed
EP-3094314-B1 TARGETED NANOCARRIERS FOR THE ADMINISTRATION OF IMMUNOSUPPRESSIVE AGENTS MUSC FOUND FOR RES DEV (US) 2021-06-23 EP disclosed
CN-108409630-B Preparation method of 3-hydroxy-2-indolone derivative in aqueous phase 宁波大学 2021-01-15 CN disclosed
CN-107686460-B Preparation method of 3-substituted-3-hydroxy-2-indolone compound 宁波大学 2020-06-12 CN disclosed
US-20200056183-A1 TARGETED NANOCARRIERS FOR THE ADMINISTRATION OF IMMUNOSUPPRESSIVE AGENTS MUSC FOUNDATION FOR RESEARCH DEVELOPMENT 2020-02-20 US disclosed
EP-2278966-B1 TREATMENT WITH OPIOID ANTAGONISTS AND MTOR INHIBITORS UNIV CHICAGO (US) 2019-10-09 EP disclosed
US-10428331-B2 Targeted nanocarriers for the administration of immunosuppressive agents MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2019-10-01 US disclosed
US-10383869-B2 Treatment with opioid antagonists and mTOR inhibitors THE UNIVERSITY OF CHICAGO (US) 2019-08-20 US disclosed
US-20110021551-A1 TREATMENT WITH OPIOID ANTAGONISTS AND mTOR INHIBITORS THE UNIVERSITY OF CHICAGO 2011-01-27 US disclosed
US-7846962-B2 3-3-di-substituted-oxindoles as inhibitors of translation initiation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-12-07 US disclosed
US-20100256388-A1 3-3-Di-Substituted-Oxindoles As Inhibitors of Translation Initiation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-10-07 US disclosed
US-20100249201-A1 3-3-Di-Substituted-Oxindoles As Inhibitors of Translation Initiation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-09-30 US disclosed
US-7737172-B2 3-3-di-substituted-oxindoles as inhibitors of translation initiation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-06-15 US disclosed
US-20090299058-A1 3-3-DI-SUBSTITUTED-OXINDOLES AS INHIBITORS OF TRANSLATION INITIATION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2009-12-03 US disclosed
WO-2009117669-A2 TREATMENT WITH OPIOID ANTAGONISTS AND MTOR INHIBITORS THE UNIVERSITY OF CHICAGO (US) 2009-09-24 WO disclosed
US-20070099976-A1 3-3-DI-SUBSTITUTED-OXINDOLES AS INHIBITORS OF TRANSLATION INITIATION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2007-05-03 US disclosed
EP-1718611-A1 3-3-DI-SUBSTITUTED-OXINDOLES AS INHIBITORS OF TRANSLATION INITIATION The President and Fellows of Harvard College (US) 2006-11-08 EP disclosed
WO-2005080335-A1 3-3-DI-SUBSTITUTED-OXINDOLES AS INHIBITORS OF TRANSLATION INITIATION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2005-09-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100256388-A1 3-3-Di-Substituted-Oxindoles As Inhibitors of Translation Initiation EIF2AK2, EIF5B, EIF4EBP1 MEN1 4058/4885KMT2A 3213/4885ALDH1A1 3721/4885
US-20090299058-A1 3-3-DI-SUBSTITUTED-OXINDOLES AS INHIBITORS OF TRANSLATION INITIATION EIF2AK2, EIF5B, EIF4EBP1 MEN1 4058/4885KMT2A 3213/4885ALDH1A1 3721/4885
US-20070099976-A1 3-3-DI-SUBSTITUTED-OXINDOLES AS INHIBITORS OF TRANSLATION INITIATION EIF2AK2, EIF5B, EIF4EBP1 MEN1 4058/4885KMT2A 3213/4885ALDH1A1 3721/4885
US-10383869-B2 Treatment with opioid antagonists and mTOR inhibitors OPRL1, OPRK1, OPRM1 MEN1 4535/4885KMT2A 1568/4885ALDH1A1 3995/4885
US-10428331-B2 Targeted nanocarriers for the administration of immunosuppressive agents CD59, CD47, CD58 MEN1 4210/4885KMT2A 4616/4885ALDH1A1 2129/4885
US-20110021551-A1 TREATMENT WITH OPIOID ANTAGONISTS AND mTOR INHIBITORS OPRL1, OPRK1, OPRM1 MEN1 4535/4885KMT2A 1568/4885ALDH1A1 3995/4885
US-20100249201-A1 3-3-Di-Substituted-Oxindoles As Inhibitors of Translation Initiation EIF2AK2, EIF5B, EIF4EBP1 MEN1 4058/4885KMT2A 3213/4885ALDH1A1 3721/4885
US-20200056183-A1 TARGETED NANOCARRIERS FOR THE ADMINISTRATION OF IMMUNOSUPPRESSIVE AGENTS CD59, CD47, CD58 MEN1 4210/4885KMT2A 4616/4885ALDH1A1 2129/4885
US-20240180894-A1 METHODS OF TREATING MENTAL AND/OR MOOD DISORDERS USING 2-BROMO-LSD ALONE OR IN COMBINATION WITH A MTOR INHIBITOR MTOR, RICTOR, RPTOR MEN1 1710/4885KMT2A 190/4885ALDH1A1 4604/4885
US-11214805-B2 Targeted nanocarriers for the administration of immunosuppressive agents CD59, CD47, CD58 MEN1 4210/4885KMT2A 4616/4885ALDH1A1 2129/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.