SCHEMBL2089449

SCHEMBL2089449

COc1ccc(-c2cc(NC(=O)CCCCN3CCCCCC3)n[nH]2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRNA3 P32297 5/20 1.00
KCNH2 Q12809 3/20 0.94
CHRNA7 P36544 1/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2055637 0.92 CHRNA3 (0.84) CHRNA3KCNH2CHRNA7
SCHEMBL1854943 0.91 KCNH2 (1.00) CHRNA3KCNH2CHRNA7
SCHEMBL2089789 0.90 KCNH2 (0.98) CHRNA3KCNH2CHRNA7
Hydrochloric Acid SCHEMBL1863445 0.90 KCNH2 (0.98) CHRNA3KCNH2CHRNA7
SCHEMBL2088367 0.90 CHRNA3 (0.81) CHRNA3KCNH2CHRNA7
Hydrochloric Acid SCHEMBL4085058 0.89 KCNH2 (0.97) CHRNA3KCNH2CHRNA7
SCHEMBL2088851 0.87 KCNH2 (1.00) CHRNA3KCNH2CHRNA7
SCHEMBL1855215 0.86 CHRNA3 (0.79) CHRNA3KCNH2CHRNA7
SCHEMBL2055604 0.83 CHRNA3 (0.72) CHRNA3KCNH2CHRNA7
SCHEMBL2090433 0.83 CHRNA3 (0.72) CHRNA3KCNH2CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163729-B2 Modulators of α7 nicotinic acetylcholine receptors and therapeutic uses thereof WYETH (US) 2012-04-24 US disclosed