SCHEMBL20904178

SCHEMBL20904178

Cc1csc(N(C)C(=O)Cc2ccc(-c3cc(F)ccc3F)cc2)n1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 8/20 0.65
CA1 P00915 8/20 0.65
CA2 P00918 8/20 0.65
CA5A P35218 8/20 0.65
CA9 Q16790 8/20 0.65
CA5B Q9Y2D0 8/20 0.65
SLC12A5 Q9H2X9 2/20 0.45
LMNA P02545 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MAPT P10636 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP2D6 P10635 1/20 0.40
WNT3A P56704 1/20 0.39
EIF4E P06730 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25892474 0.92 CA12 (0.55) CA12CA1CA2CA5ACA9
SCHEMBL25892626 0.90 CA12 (0.53) CA12CA1CA2CA5ACA9
SCHEMBL24767415 0.88 CA12 (0.61) CA12CA1CA2CA5ACA9
SCHEMBL20888475 0.87 CA12 (0.64) CA12CA1CA2CA5ACA9
SCHEMBL25893787 0.87 CA12 (0.59) CA12CA1CA2CA5ACA9
SCHEMBL25894205 0.85 CA12 (0.58) CA12CA1CA2CA5ACA9
SCHEMBL24767096 0.81 CA12 (0.74) CA12CA1CA2CA5ACA9
SCHEMBL22427646 0.81 CA12 (0.73) CA12CA1CA2CA5ACA9
SCHEMBL31187475 0.80 CA12 (0.72) CA12CA1CA2CA5ACA9
SCHEMBL20876170 0.80 CA12 (0.72) CA12CA1CA2CA5ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023135303-A1 SOLID CRYSTALLINE FORMS OF HELICASE-PRIMASE INHIBITORS AND PROCESS OF PREPARATION THEREOF INNOVATIVE MOLECULES GMBH (DE) 2023-07-20 WO disclosed
EP-4209491-A1 ENANTIOMERS OF SUBSTITUTED THIAZOLES AS ANTIVIRAL COMPOUNDS Innovative Molecules GmbH (DE) 2023-07-12 EP disclosed
EP-3692039-B1 ENANTIOMERS OF SUBSTITUTED THIAZOLES AS ANTIVIRAL COMPOUNDS INNOVATIVE MOLECULES GMBH (DE) 2022-12-14 EP disclosed
CN-109071473-B Antiviral compounds 创新分子股份有限公司 2022-12-09 CN disclosed
EP-3440063-B1 AMINOTHIAZOLE DERIVATIVES USEFUL AS ANTIVIRAL AGENTS INNOVATIVE MOLECULES GMBH (DE) 2020-08-05 EP disclosed
EP-3440063-B1 AMINOTHIAZOLE DERIVATIVES USEFUL AS ANTIVIRAL AGENTS INNOVATIVE MOLECULES GMBH (DE) 2020-08-05 EP disclosed
WO-2020109389-A1 HELICASE PRIMASE INHIBITORS FOR TREATING CANCER IN A COMBINATION THERAPY WITH ONCOLYTIC VIRUSES INNOVATIVE MOLECULES GMBH (DE) 2020-06-04 WO disclosed
US-20200148652-A1 Aminothiazole Derivatives Useful As Antiviral Agents INNOVATIVE MOLECULES GMBH (DE) 2020-05-14 US disclosed
US-20200148652-A1 Aminothiazole Derivatives Useful As Antiviral Agents INNOVATIVE MOLECULES GMBH (DE) 2020-05-14 US disclosed
US-10590094-B2 Aminothiazole derivatives useful as antiviral agents INNOVATIVE MOLECULES GMBH (DE) 2020-03-17 US disclosed
US-20190112285-A1 Aminothiazole Derivatives Useful As Antiviral Agents INNOVATIVE MOLECULES GMBH (DE) 2019-04-18 US disclosed
CN-109071473-A Novel antivirus compound 创新分子股份有限公司 2018-12-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200148652-A1 Aminothiazole Derivatives Useful As Antiviral Agents MAVS, EIF2AK2, SARS1 CA12 4742/4885CA1 4843/4885CA2 4245/4885
US-20190112285-A1 Aminothiazole Derivatives Useful As Antiviral Agents MAVS, EIF2AK2, SARS1 CA12 4770/4885CA1 4844/4885CA2 4253/4885
US-10590094-B2 Aminothiazole derivatives useful as antiviral agents MAVS, EIF2AK2, SARS1 CA12 4770/4885CA1 4844/4885CA2 4253/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.