SCHEMBL20904188

SCHEMBL20904188

CC(C)N(C)C(=O)Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC4 O15439 1/20 0.55
LMNA P02545 1/20 0.55
GAA P10253 1/20 0.55
TSHR P16473 1/20 0.55
PTGS1 P23219 1/20 0.55
HTT P42858 1/20 0.55
ALDH1A1 P00352 2/20 0.51
HPGD P15428 2/20 0.51
MAPT P10636 1/20 0.51
NPY5R Q15761 1/20 0.50
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA5A P35218 2/20 0.48
CA9 Q16790 2/20 0.48
CA5B Q9Y2D0 2/20 0.48
USP30 Q70CQ3 1/20 0.48
KMT2A Q03164 2/20 0.46
CCR5 P51681 1/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5053649 0.90 TSHR (0.52) TSHRHPGDNPY5RKMT2AMEN1
SCHEMBL20888587 0.82 LMNA (0.62) ABCC4LMNAGAATSHRPTGS1
SCHEMBL20904187 0.82 NPSR1 (0.55) ALDH1A1MAPTNPY5RCA12CA1
SCHEMBL20904180 0.81 CA12 (0.55) NPY5RCA12CA1CA2CA5A
SCHEMBL12856883 0.77 NPY5R (0.54) GAATSHRNPY5RKMT2AMEN1
SCHEMBL1515926 0.77 LMNA (0.55) ABCC4LMNAGAATSHRPTGS1
SCHEMBL5966848 0.76 TSHR (0.50) TSHRNPY5RKMT2AMEN1
SCHEMBL2625190 0.75 LMNA (0.62) ABCC4LMNAGAATSHRPTGS1
SCHEMBL20904160 0.74 CA12 (0.55) NPY5RCA12CA1CA2CA5A
Felbinac SCHEMBL384892 0.74 LMNA (0.95) ABCC4LMNAGAATSHRPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200289486-A1 Enantiomers Of Substituted Thiazoles As Antiviral Compounds INNOVATIVE MOLECULES GMBH (DE) 2020-09-17 US disclosed
US-20200148652-A1 Aminothiazole Derivatives Useful As Antiviral Agents INNOVATIVE MOLECULES GMBH (DE) 2020-05-14 US disclosed
US-10590094-B2 Aminothiazole derivatives useful as antiviral agents INNOVATIVE MOLECULES GMBH (DE) 2020-03-17 US disclosed
US-20190112285-A1 Aminothiazole Derivatives Useful As Antiviral Agents INNOVATIVE MOLECULES GMBH (DE) 2019-04-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200148652-A1 Aminothiazole Derivatives Useful As Antiviral Agents MAVS, EIF2AK2, SARS1 ABCC4 2595/4885LMNA 4099/4885GAA 710/4885
US-20190112285-A1 Aminothiazole Derivatives Useful As Antiviral Agents MAVS, EIF2AK2, SARS1 ABCC4 2433/4885LMNA 4100/4885GAA 665/4885
US-20200289486-A1 Enantiomers Of Substituted Thiazoles As Antiviral Compounds EIF2AK2, MAVS, ZC3HAV1 ABCC4 1287/4885LMNA 3312/4885GAA 416/4885
US-10590094-B2 Aminothiazole derivatives useful as antiviral agents MAVS, EIF2AK2, SARS1 ABCC4 2433/4885LMNA 4100/4885GAA 665/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.