SCHEMBL20908006

SCHEMBL20908006

C[C@H](COC(=O)NC1CC1)c1ccc(Cl)c(C(N)=O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.39
SLC6A3 Q01959 2/20 0.39
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TSHR P16473 2/20 0.38
PRCP P42785 1/20 0.37
LMNA P02545 1/20 0.37
DPP4 P27487 1/20 0.37
DPP7 Q9UHL4 1/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
DRD2 P14416 1/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20899815 0.87 DPP4 (0.39) HSP90AA1SLC6A3NPSR1TSHRLMNA
SCHEMBL20899715 0.87 DPP4 (0.39) HSP90AA1SLC6A3NPSR1TSHRLMNA
SCHEMBL28407779 0.84 TSHR (0.37) HSP90AA1SLC6A3NPSR1TSHRPRCP
SCHEMBL28407777 0.84 TSHR (0.37) HSP90AA1SLC6A3NPSR1TSHRPRCP
SCHEMBL21112408 0.84 TSHR (0.38) HSP90AA1SLC6A3NPSR1TSHRLMNA
SCHEMBL20899810 0.84 TSHR (0.38) HSP90AA1SLC6A3NPSR1TSHRLMNA
SCHEMBL21112802 0.81 BTK (0.39) KMT2ADRD2HPGDKDM4EALDH1A1
SCHEMBL29640289 0.81 BTK (0.39) KMT2ADRD2HPGDKDM4EALDH1A1
SCHEMBL20907825 0.81 BTK (0.39) KMT2ADRD2HPGDKDM4EALDH1A1
SCHEMBL20899811 0.76 LMNA (0.36) HSP90AA1SLC6A3NPSR1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019075291-A1 1-BENZYL-2-IMINO-4-PHENYL-5-OXOIMIDAZOLIDINE DERIVATIVES AS HIV PROTEASE INHIBITORS GILEAD SCIENCES, INC. (US) 2019-04-18 WO disclosed