SCHEMBL20909684

SCHEMBL20909684

Cc1ccc2c(N(C)C)noc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.39
HTR3A P46098 2/20 0.39
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
LMNA P02545 3/20 0.38
KDM4E B2RXH2 2/20 0.38
TP53 P04637 1/20 0.36
ESR1 P03372 4/20 0.36
ESR2 Q92731 4/20 0.36
GAA P10253 3/20 0.35
APP P05067 1/20 0.35
MAOB P27338 1/20 0.34
RECQL P46063 1/20 0.34
KMT2A Q03164 1/20 0.34
HPGD P15428 1/20 0.33
HTR2A P28223 1/20 0.33
DRD3 P35462 1/20 0.33
CYP1A2 P05177 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20883957 0.77 TSHR (0.35) ALDH1A1KDM4EESR1ESR2KMT2A
SCHEMBL20884969 0.77 TBK1 (0.34) ALDH1A1MAPTLMNAKDM4ETP53
SCHEMBL4399692 0.76 CHRNB2 (0.45) CHRNA7HTR3AALDH1A1MAPTKDM4E
SCHEMBL20439174 0.75 HIF1A (0.44) ALDH1A1LMNAESR1ESR2GAA
SCHEMBL23474002 0.73 MAPT (0.42) CHRNA7HTR3AALDH1A1MAPTLMNA
SCHEMBL8233882 0.73 F9 (0.47) CHRNA7HTR3AALDH1A1MAPTLMNA
SCHEMBL25591522 0.73 CHRNA7 (0.40) CHRNA7HTR3AALDH1A1MAPTLMNA
SCHEMBL1101176 0.73 ESR1 (0.45) CHRNA7HTR3AMAPTESR1ESR2
SCHEMBL16048336 0.72 CSF1R (0.39)
SCHEMBL23175518 0.71 HTR2A (0.51) CHRNA7HTR3AHTR2ADRD3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019074979-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF GIRAFPHARMA, LLC (US) 2019-04-18 WO disclosed