SCHEMBL209177

SCHEMBL209177

CNC(c1ccccc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.52
RAB9A P51151 1/20 0.52
GRM7 Q14831 1/20 0.52
TSHR P16473 4/20 0.50
HTR2A P28223 3/20 0.50
CYP3A4 P08684 2/20 0.50
ALOX15 P16050 2/20 0.50
CHRM2 P08172 1/20 0.50
ADRA1A P35348 1/20 0.50
RGS12 O14924 1/20 0.50
GLA P06280 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
PKM P14618 1/20 0.50
ALOX12 P18054 1/20 0.50
ADRA2C P18825 1/20 0.50
NFKB1 P19838 1/20 0.50
CYP2C19 P33261 1/20 0.50
THPO P40225 1/20 0.50
GNAI1 P63096 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2254912 0.97 TSHR (0.54) MTORRAB9AGRM7TSHRHTR2A
SCHEMBL13184555 0.88 LMNA (0.56) MTORRAB9AGRM7TSHRHTR2A
Acetonitrile SCHEMBL27872054 0.88 MTOR (0.43) MTORRAB9AGRM7TSHRHTR2A
Acetic Acid SCHEMBL9853096 0.88 LMNA (0.47) MTORRAB9AGRM7TSHRHTR2A
SCHEMBL29266047 0.88 LMNA (0.56) MTORRAB9AGRM7TSHRHTR2A
SCHEMBL23209633 0.86 ALDH1A1 (0.46) MTORRAB9AGRM7TSHRHTR2A
SCHEMBL4759648 0.86 SLC6A4 (0.50) TSHRCHRM2ADRA1ACYP2D6CYP2C19
SCHEMBL1038300 0.86 SLC6A2 (0.58) MTORRAB9AGRM7TSHRHTR2A
Hydrochloric Acid SCHEMBL29091952 0.86 LMNA (0.55) MTORRAB9AGRM7TSHRHTR2A
Hydrochloric Acid SCHEMBL31250027 0.84 IDO1 (0.50) TSHRCYP3A4ALOX15CHRM2ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2568 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250352656-A1 SYNTHETIC CATIONIC PEPTIDOMIMETICS, THEIR DERIVATIVES AND PREPARATION THEREOF ALONG WITH COMPOSITIONS FOR VARIOUS MEDICAL APPLICATIONS PEPTOMER THERAPEUTICS PRIVATE LTD (IN) 2025-11-20 US claimed
EP-4525827-A1 SYNTHETIC CATIONIC PEPTIDOMIMETICS, THEIR DERIVATIVES AND PREPARATION THEREOF ALONG WITH COMPOSITIONS FOR VARIOUS MEDICAL APPLICATIONS Peptomer Therapeutics Private Limited (IN) 2025-03-26 EP claimed
CN-114409493-B Method for synthesizing 9-aryl fluorene compound 浙江工业大学 2024-02-23 CN claimed
WO-2023209728-A1 SYNTHETIC CATIONIC PEPTIDOMIMETICS, THEIR DERIVATIVES AND PREPARATION THEREOF ALONG WITH COMPOSITIONS FOR VARIOUS MEDICAL APPLICATIONS PEPTOMER THERAPEUTICS PRIVATE LIMITED (IN) 2023-11-02 WO claimed
US-20210163541-A1 Method for Preparing PNA Oligomer SEASUNBIO MATERIALS (KR) 2021-06-03 US claimed
EP-3110828-B1 CONTINUOUS FLOW PEPTIDE SYNTHESIS UNIV SZEGEDI (HU) 2020-12-09 EP claimed
CN-110669058-A Tricyclic quinolone carboxylic acid and preparation method thereof 江西农业大学 2020-01-10 CN claimed
EP-3110828-A1 CONTINUOUS FLOW PEPTIDE SYNTHESIS Szegedi Tudományegyetem (HU) 2017-01-04 EP claimed
WO-2015128687-A1 CONTINUOUS FLOW PEPTIDE SYNTHESIS Szegedi Tudományegyetem (HU) 2015-09-03 WO claimed
US-20130274440-A1 DIMEDON DERIVATIVE AND A METHOD FOR THE PURIFICATION OF PNA AND PEPTIDE OLIGOMERS DEUTSCHES KREBSFORSCHUNGSZENTRUM (DE) 2013-10-17 US claimed
WO-1991007429-A1 ANTI-AGGREGATORY PEPTIDES CONTAINING A MERCAPTAN OR SULFIDE MOIETY SMITHKLINE BEECHAM CORPORATION (US) 1991-05-30 WO claimed
EP-0408371-A1 Hemoregulatory peptides SMITHKLINE BEECHAM CORPORATION (US) 1991-01-16 EP claimed
EP-0376218-A2 Racemization free attachment of amino acids to solid phase PERSEPTIVE BIOSYSTEMS, INC. (US) 1990-07-04 EP claimed
EP-0348819-A2 Anorexigenic and hypotensive peptides ZAMBON GROUP S.p.A. (IT) 1990-01-03 EP claimed
EP-0341915-A2 Anti-aggregatory peptides SMITHKLINE BEECHAM CORPORATION (US) 1989-11-15 EP claimed
EP-0341935-A2 A solid phase process for synthesizing Thymosin alpha 1 ALPHA-1 BIOMEDICALS, INC. (US) 1989-11-15 EP claimed
US-4855407-A Solid phase process for synthesizing peptides ALPHA-1 BIOMEDICALS, INC. (US) 1989-08-08 US claimed
EP-0315367-A2 Polypeptides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-10 EP claimed
EP-0200404-A2 Solid phase process for synthesizing peptides ALPHA-1 BIOMEDICALS, INC. (US) 1986-11-05 EP claimed
EP-0021620-B1 WATER-SOLUBLE PEPTIDES AFFECTING GONADAL FUNCTION THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 1983-02-23 EP claimed