Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | MEN1 | O00255 | 11/20 | 0.72 |
| ▸ | KMT2A | Q03164 | 11/20 | 0.72 |
| ▸ | ALDH1A1 | P00352 | 9/20 | 0.72 |
| ▸ | MAPT | P10636 | 9/20 | 0.72 |
| ▸ | MCL1 | Q07820 | 8/20 | 0.72 |
| ▸ | HPGD | P15428 | 7/20 | 0.72 |
| ▸ | KDM4E | B2RXH2 | 7/20 | 0.72 |
| ▸ | L3MBTL1 | Q9Y468 | 7/20 | 0.72 |
| ▸ | BLM | P54132 | 6/20 | 0.72 |
| ▸ | THRB | P10828 | 6/20 | 0.72 |
| ▸ | PKM | P14618 | 6/20 | 0.72 |
| ▸ | RECQL | P46063 | 5/20 | 0.72 |
| ▸ | TDP1 | Q9NUW8 | 5/20 | 0.72 |
| ▸ | NR4A1 | P22736 | 4/20 | 0.72 |
| ▸ | ALOX12 | P18054 | 3/20 | 0.72 |
| ▸ | BID | P55957 | 1/20 | 0.72 |
| ▸ | BCL2A1 | Q16548 | 1/20 | 0.72 |
| ▸ | POLB | P06746 | 9/20 | 0.64 |
| ▸ | HTT | P42858 | 3/20 | 0.64 |
| ▸ | APEX1 | P27695 | 3/20 | 0.64 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL30518187 | 1.00 | MEN1 (0.72) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL13856422 | 0.84 | MEN1 (1.00) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL6722302 | 0.82 | MCL1 (0.77) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL24277667 | 0.80 | MCL1 (1.00) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL26294531 | 0.80 | MEN1 (0.76) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL13856429 | 0.78 | MEN1 (1.00) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL15814086 | 0.78 | MEN1 (0.84) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL2113647 | 0.78 | ALDH1A1 (1.00) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL26293058 | 0.78 | MEN1 (0.78) | MEN1KMT2AALDH1A1MAPTMCL1 | |
| SCHEMBL26294069 | 0.77 | MEN1 (0.68) | MEN1KMT2AALDH1A1MAPTMCL1 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-20230233501-A1 | COMPOSITIONS FOR INHIBITING 3' REPAIR EXONUCLEASE 2 AND METHODS OF SCREENING FOR SUCH COMPOSITIONS | UNIV TEXAS (US) | 2023-07-27 | — | — | US | claimed |
| US-20200253913-A1 | COMPOSITIONS FOR INHIBITING 3' REPAIR EXONUCLEASE 2 AND METHODS OF SCREENING FOR SUCH COMPOSITIONS | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2020-08-13 | — | — | US | claimed |
| US-20200239969-A1 | METHODS AND COMPOSITIONS FOR USE OF TREX2 AS DIAGNOSTIC AND PROGNOSTIC MARKER FOR CANCER | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2020-07-30 | — | — | US | claimed |
| WO-2019079222-A1 | COMPOSITIONS FOR INHIBITING 3' REPAIR EXONUCLEASE 2 AND METHODS OF SCREENING FOR SUCH COMPOSITIONS | BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) | 2019-04-25 | — | — | WO | claimed |
| WO-2019079255-A1 | METHODS AND COMPOSITIONS FOR USE OF TREX2 AS DIAGNOSTIC AND PROGNOSTIC MARKER FOR CANCER | BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) | 2019-04-25 | — | — | WO | claimed |
| US-20230233501-A1 | COMPOSITIONS FOR INHIBITING 3' REPAIR EXONUCLEASE 2 AND METHODS OF SCREENING FOR SUCH COMPOSITIONS | UNIV TEXAS (US) | 2023-07-27 | — | — | US | disclosed |
| US-11612580-B2 | Compositions for inhibiting 3′ repair exonuclease 2 and methods of screening for such compositions | THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) | 2023-03-28 | — | — | US | disclosed |
| US-20200253913-A1 | COMPOSITIONS FOR INHIBITING 3' REPAIR EXONUCLEASE 2 AND METHODS OF SCREENING FOR SUCH COMPOSITIONS | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2020-08-13 | — | — | US | disclosed |
| US-20200239969-A1 | METHODS AND COMPOSITIONS FOR USE OF TREX2 AS DIAGNOSTIC AND PROGNOSTIC MARKER FOR CANCER | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2020-07-30 | — | — | US | disclosed |
| WO-2019079222-A1 | COMPOSITIONS FOR INHIBITING 3' REPAIR EXONUCLEASE 2 AND METHODS OF SCREENING FOR SUCH COMPOSITIONS | BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) | 2019-04-25 | — | — | WO | disclosed |
| WO-2019079255-A1 | METHODS AND COMPOSITIONS FOR USE OF TREX2 AS DIAGNOSTIC AND PROGNOSTIC MARKER FOR CANCER | BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) | 2019-04-25 | — | — | WO | disclosed |