SCHEMBL20920125

SCHEMBL20920125

O=[N+]([O-])c1ccc2[nH]c3ccc(Br)cc3c2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.59
GABRG2 P18507 1/20 0.59
GABRB3 P28472 1/20 0.59
GABRA5 P31644 1/20 0.59
GABRA2 P47869 1/20 0.59
CTSV O60911 2/20 0.58
CTSL P07711 2/20 0.58
PARP1 P09874 2/20 0.58
CDK5 Q00535 3/20 0.57
CDK5R1 Q15078 3/20 0.57
CA12 O43570 2/20 0.57
CA9 Q16790 2/20 0.57
KIF11 P52732 1/20 0.56
CCNB2 O95067 1/20 0.53
CDK1 P06493 1/20 0.53
CCNB1 P14635 1/20 0.53
GSK3B P49841 1/20 0.53
CCNB3 Q8WWL7 1/20 0.53
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21828647 0.92 CTSV (0.70) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL155013 0.89 GABRA1 (0.70) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL29540314 0.89 GABRA1 (0.70) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL30272743 0.81 CTSV (0.79) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL30272742 0.81 CTSV (0.79) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL30272741 0.81 CTSV (0.79) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL151534 0.81 CTSV (0.79) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL12722533 0.79 MAPT (0.59) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL17396637 0.79 GABRA1 (0.59) GABRA1GABRG2GABRB3GABRA5GABRA2
SCHEMBL30272747 0.79 GABRA1 (0.59) GABRA1GABRG2GABRB3GABRA5GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019076336-A1 PYRAZOLYL-CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF 江苏豪森药业集团有限公司 2019-04-25 WO disclosed