SCHEMBL20923256

SCHEMBL20923256

N#Cc1cc(-c2ccccc2)c(-n2c3ccc(-c4cc(C(F)(F)F)cc(C(F)(F)F)c4)cc3c3cc(-c4cc(C(F)(F)F)cc(C(F)(F)F)c4)ccc32)cc1-c1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.37
GPBAR1 Q8TDU6 4/20 0.36
METAP2 P50579 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
EPHX2 P34913 1/20 0.34
ICMT O60725 1/20 0.34
PRKACA P17612 1/20 0.33
CDK8 P49336 1/20 0.33
CLK2 P49760 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CDK9 P50750 1/20 0.33
CDK5 Q00535 1/20 0.33
PRKCQ Q04759 1/20 0.33
ROCK1 Q13464 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20923770 0.97 METAP2 (0.36) PIK3CAGPBAR1METAP2CYP11B1CYP11B2
SCHEMBL20923601 0.96 GPBAR1 (0.36) PIK3CAGPBAR1METAP2CYP11B1CYP11B2
SCHEMBL20923847 0.93 METAP2 (0.36) PIK3CAGPBAR1METAP2CYP11B1CYP11B2
SCHEMBL20923768 0.92 METAP2 (0.37) PIK3CAGPBAR1METAP2CYP11B1CYP11B2
SCHEMBL20923274 0.92 METAP2 (0.36) PIK3CAGPBAR1METAP2CYP11B1CYP11B2
SCHEMBL19908956 0.91 METAP2 (0.38) GPBAR1METAP2CYP11B1CYP11B2EPHX2
SCHEMBL19919458 0.90 CYP11B1 (0.35) GPBAR1METAP2CYP11B1CYP11B2EPHX2
SCHEMBL22170431 0.90 METAP2 (0.37) GPBAR1METAP2CYP11B1CYP11B2EPHX2
SCHEMBL20923121 0.90 CYP19A1 (0.38) GPBAR1METAP2CYP11B1CYP11B2ALDH1A1
SCHEMBL19919686 0.90 CYP11B1 (0.37) GPBAR1METAP2CYP11B1CYP11B2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3266772-B1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2019-04-24 EP disclosed