SCHEMBL20925129

SCHEMBL20925129

C=CC(=O)OCc1ccc(-c2ccc(OC(=O)C=C)c(F)c2)cc1F

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
THRB P10828 3/20 0.35
THRA P10827 1/20 0.35
NAAA Q02083 6/20 0.34
CTSK P43235 1/20 0.33
ERN1 O75460 1/20 0.33
ALDH1A1 P00352 2/20 0.33
TP53 P04637 2/20 0.33
HIF1A Q16665 2/20 0.33
HSD17B10 Q99714 1/20 0.33
FAAH O00519 1/20 0.32
ESR1 P03372 2/20 0.32
ESR2 Q92731 2/20 0.32
FFAR1 O14842 2/20 0.32
PPARD Q03181 2/20 0.32
TYMS P04818 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13967526 0.89 NAAA (0.33) TSHRPOLBMAPK1NAAACTSK
SCHEMBL18511256 0.88 NAAA (0.38) THRBTHRANAAAERN1FAAH
SCHEMBL16977650 0.88 THRB (0.41) TSHRTHRBNAAAALDH1A1TP53
SCHEMBL16977640 0.87 THRB (0.38) TSHRPOLBMAPK1THRBERN1
SCHEMBL9607776 0.86 ERN1 (0.40) TSHRPOLBMAPK1THRBTHRA
SCHEMBL15338873 0.81 THRB (0.36) TSHRTHRBTHRAALDH1A1TP53
SCHEMBL20174163 0.81 NPC1 (0.36) TSHRPOLBMAPK1ERN1FAAH
SCHEMBL2604655 0.80 TYMS (0.41) TSHRPOLBMAPK1THRBTHRA
SCHEMBL9613625 0.80 THRB (0.43) TSHRPOLBMAPK1THRBTHRA
SCHEMBL14984569 0.80 POLB (0.38) TSHRPOLBMAPK1THRBTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3234689-B1 LIGHT MODULATION ELEMENT MERCK PATENT GMBH (DE) 2020-01-29 EP disclosed
EP-3067406-B1 LIQUID CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2019-04-24 EP disclosed