SCHEMBL20928233

SCHEMBL20928233

Cc1ccc(C)c2ncc(I)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TET2 Q6N021 4/20 0.39
CCR1 P32246 3/20 0.39
CCR5 P51681 3/20 0.39
CCR8 P51685 3/20 0.39
ALDH1A1 P00352 3/20 0.36
IDO1 P14902 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
GLA P06280 1/20 0.33
PKM P14618 1/20 0.33
PSMD14 O00487 1/20 0.32
COPS5 Q92905 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTT P42858 1/20 0.32
CYP1A2 P05177 1/20 0.32
USP2 O75604 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22326639 0.85 TET2 (0.56) TET2CCR1CCR5CCR8IDO1
SCHEMBL20928236 0.78 CCR1 (0.52) CCR1CCR5CCR8ALDH1A1MEN1
SCHEMBL23763291 0.72 CCR1 (0.38) TET2CCR1CCR5CCR8SMN1; SMN2
SCHEMBL21064338 0.72 CYP1A2 (0.39) ALDH1A1KDM4ECYP1A2NPC1
SCHEMBL24121697 0.72 CCR1 (0.42) TET2CCR1CCR5CCR8IDO1
SCHEMBL13486493 0.72 KDM4E (0.44) CCR1CCR5CCR8ALDH1A1MEN1
SCHEMBL25191210 0.70 IDO1 (0.41) TET2CCR1CCR5CCR8IDO1
SCHEMBL22326650 0.69 CCR1 (0.42) TET2CCR1CCR5CCR8KDM4E
SCHEMBL7681923 0.69 ALDH1A1 (0.45) ALDH1A1MEN1KMT2AKDM4EL3MBTL1
SCHEMBL17423371 0.67 ALDH1A1 (0.52) CCR1CCR5CCR8ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019076343-A1 PD-1/PD-L1 SMALL-MOLECULE INHIBITOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海长森药业有限公司 2019-04-25 WO disclosed