SCHEMBL20928236

SCHEMBL20928236

Cc1cnc2c(C)ccc(C)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.52
CCR5 P51681 5/20 0.52
CCR8 P51685 5/20 0.52
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
KDM4E B2RXH2 3/20 0.41
PSMD14 O00487 2/20 0.41
COPS5 Q92905 2/20 0.41
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 3/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PARP1 P09874 2/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CYP2A6 P11509 1/20 0.34
SLC6A2 P23975 1/20 0.34
HTT P42858 1/20 0.34
GLA P06280 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22326640 0.84 CCR1 (0.45) CCR1CCR5CCR8NOS3NOS1
SCHEMBL24916307 0.81 CCR1 (0.42) CCR1CCR5CCR8PKM
SCHEMBL20928233 0.78 TET2 (0.39) CCR1CCR5CCR8KDM4EPSMD14
SCHEMBL5226896 0.73 CCR1 (0.52) CCR1CCR5CCR8NOS3NOS1
SCHEMBL6174019 0.73 CYP2A6 (0.46) CCR1CCR5CCR8KDM4ESMN1; SMN2
SCHEMBL7681923 0.72 ALDH1A1 (0.45) KDM4EPSMD14ALDH1A1CYP1A2MEN1
SCHEMBL18644122 0.72 CCR1 (0.42) CCR1CCR5CCR8NOS3NOS1
SCHEMBL11920831 0.72 KDM4E (0.44) CCR1CCR5CCR8NOS3NOS1
SCHEMBL29430432 0.72 CCR1 (0.57) CCR1CCR5CCR8NOS3NOS1
SCHEMBL22615073 0.72 CCR1 (0.57) CCR1CCR5CCR8NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019076343-A1 PD-1/PD-L1 SMALL-MOLECULE INHIBITOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海长森药业有限公司 2019-04-25 WO disclosed