SCHEMBL20934880

SCHEMBL20934880

Nc1ccc(NCCNC2COC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.39
MAPT P10636 3/20 0.35
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
GAA P10253 2/20 0.32
PTH1R Q03431 1/20 0.32
EPHX1 P07099 1/20 0.31
RAB9A P51151 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX12 P18054 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MAP4K4 O95819 1/20 0.30
KDM1A O60341 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24375404 0.83 PTH1R (0.33) MAPTPTH1RMAP4K4
SCHEMBL20934767 0.83 FPR2 (0.37) MAPTGAARAB9AALDH1A1L3MBTL1
SCHEMBL180817 0.77 APP (0.55) APPMAPTMAOAMAOBGAA
Hydrochloric Acid SCHEMBL4952599 0.74 APP (0.53) APPMAPTMAOAMAOBGAA
SCHEMBL24030297 0.74 DDB1 (0.39) APPMAPTGAAEPHX1RAB9A
SCHEMBL20934859 0.73 MAPT (0.37) MAPTPTH1RALDH1A1
SCHEMBL5155907 0.71 APP (0.50) APPMAPTMAOAMAOBGAA
Hydrochloric Acid SCHEMBL5467007 0.69 APP (0.48) APPMAPTMAOAMAOBGAA
SCHEMBL2024986 0.68 MAPT (0.56) APPMAPTMAOAMAOBRAB9A
SCHEMBL34107 0.68 PRSS1 (0.54) APPMAPTMAOAMAOBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019079373-A1 PYRIMIDINE TBK/IKKε INHIBITOR COMPOUNDS AND USES THEREOF MERCK PATENT GMBH (DE) 2019-04-25 WO disclosed