SCHEMBL20934767

SCHEMBL20934767

Brc1ccc(NCCNC2COC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 1/20 0.37
MAPT P10636 4/20 0.35
AGER Q15109 1/20 0.35
POLB P06746 1/20 0.34
DRD2 P14416 2/20 0.33
DRD3 P35462 2/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
KMT2A Q03164 6/20 0.33
MEN1 O00255 5/20 0.33
LMNA P02545 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
GAA P10253 4/20 0.33
RAB9A P51151 4/20 0.33
NPC1 O15118 3/20 0.33
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20934880 0.83 APP (0.39) MAPTL3MBTL1ALDH1A1GAARAB9A
SCHEMBL11531629 0.77 MAPT (0.55) MAPTAGERKMT2AMEN1LMNA
SCHEMBL24375404 0.76 PTH1R (0.33) MAPTDRD2DRD3DRD4
SCHEMBL22864457 0.74 FPR2 (0.42) FPR2POLBKMT2AMEN1LMNA
SCHEMBL20934859 0.73 MAPT (0.37) MAPTALDH1A1
SCHEMBL30314739 0.71 AGER (0.45) MAPTAGERDRD2DRD3DRD1
SCHEMBL24123583 0.66 MAPT (0.65) MAPTPOLBKMT2AMEN1L3MBTL1
SCHEMBL1947781 0.65 AGER (0.44) MAPTAGERKMT2AMEN1LMNA
SCHEMBL1554174 0.65 CYP1A2 (0.53) MAPTAGERKMT2AMEN1LMNA
SCHEMBL3041532 0.65 AGER (0.48) FPR2MAPTAGERKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019079373-A1 PYRIMIDINE TBK/IKKε INHIBITOR COMPOUNDS AND USES THEREOF MERCK PATENT GMBH (DE) 2019-04-25 WO disclosed