SCHEMBL2097440

SCHEMBL2097440

Nc1nc2nc[nH]c2c(=O)n1-c1cc(Br)cs1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGMT P16455 3/20 0.47
PNP P00491 1/20 0.39
DPP4 P27487 1/20 0.37
PIN1 Q13526 1/20 0.36
PDPK1 O15530 1/20 0.36
GDA Q9Y2T3 1/20 0.36
BRAF P15056 1/20 0.35
CDK2 P24941 3/20 0.34
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
CDK1 P06493 2/20 0.33
CCNB1 P14635 2/20 0.33
CCNA2 P20248 2/20 0.33
CCNA1 P78396 2/20 0.33
GRIA1 P42261 1/20 0.32
GRIA2 P42262 1/20 0.32
GRIA3 P42263 1/20 0.32
GRIA4 P48058 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2097431 0.81 MGMT (0.36) MGMTPNPPDPK1
SCHEMBL3310029 0.78 HCAR1 (0.46) PNPDPP4PIN1PDPK1GDA
SCHEMBL5084763 0.78 MGMT (0.52) MGMTPNPDPP4PIN1PDPK1
SCHEMBL1286947 0.72 MAPK1 (0.51) MGMTPNPDPP4PIN1CDK2
SCHEMBL11610799 0.72 DPP4 (0.44) PNPDPP4PIN1PDPK1GDA
Hydrochloric Acid SCHEMBL21799343 0.71 MAPK1 (0.50) MGMTPNPDPP4PIN1CDK2
SCHEMBL41788 0.70 PNP (0.50) MGMTPNPDPP4PDPK1GDA
SCHEMBL1286944 0.70 PNP (0.38) PNPDPP4ALDH1A1
SCHEMBL28106050 0.70 ATAD2 (0.39) MGMTPNPDPP4CYP1A2CYP2C19
SCHEMBL20579 0.69 DPP4 (0.50) MGMTPNPDPP4PDPK1GDA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730298-B1 SPECIFIC SUBSTRATES FOR O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE EPFL ECOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (CH) 2015-11-11 EP disclosed
US-8163479-B2 Specific substrates for O6-alkylguanine-DNA alkyltransferase ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2012-04-24 US disclosed