SCHEMBL209789

SCHEMBL209789

Cn1cncc1CN1CCN(C(=O)O)CC1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
FNTA P49354 2/20 0.39
FNTB P49356 2/20 0.39
PGGT1B P53609 1/20 0.39
GRM2 Q14416 1/20 0.37
OPRM1 P35372 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
CHRM5 P08912 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
MLNR O43193 1/20 0.36
PLA2G7 Q13093 1/20 0.36
MGLL Q99685 1/20 0.36
ABHD6 Q9BV23 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16538615 0.76 CHRM5 (0.38) MEN1KMT2ACHRM5KDM4EMLNR
SCHEMBL15473910 0.75 CHKA (0.49) KDM4EALDH1A1POLB
SCHEMBL12424288 0.73 ALDH1A1 (0.45) CHRM5ALDH1A1
SCHEMBL210157 0.71 ALDH1A1 (0.48) MEN1KMT2AKDM4EALDH1A1POLB
SCHEMBL7665146 0.71 FNTA (0.73) FNTAFNTBPGGT1B
SCHEMBL209854 0.71 ARG1 (0.42) KDM4EALDH1A1
SCHEMBL18923901 0.71 PIK3CD (0.36) FNTAFNTBOPRM1CHRM5ALDH1A1
SCHEMBL210854 0.70 ALDH1A1 (0.40) MEN1KMT2AOPRM1KDM4EALDH1A1
SCHEMBL12384834 0.70 TLR9 (0.39) MEN1KMT2ACHRM5KDM4E
SCHEMBL20458924 0.70 CXCR4 (0.47) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963315-B1 ENZYME INHIBITORS CANCER REC TECH LTD (GB) 2014-10-08 EP disclosed
US-8088761-B2 Enzyme inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2012-01-03 US disclosed
US-20090247507-A1 Enzyme Inhibitors THE INSTITUTE OF CANCER RESEARCH (GB) 2009-10-01 US disclosed
EP-1963315-A2 ENZYME INHIBITORS The Institute of Cancer Research (GB) 2008-09-03 EP disclosed
WO-2007072017-A2 ENZYME INHIBITORS THE INSTITUTE OF CANCER RESEARCH (GB) 2007-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090247507-A1 Enzyme Inhibitors AURKC, AURKB, AURKA MEN1 471/4885KMT2A 384/4885FNTA 2235/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.