SCHEMBL2098052

SCHEMBL2098052

CN(C)c1ccc(N=Nc2ccc(C(=O)NCCCn3cnc4c(OCc5ccc(CNC(=O)C(F)(F)F)cc5)nc(N)nc43)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.42
HDAC1 Q13547 14/20 0.41
HDAC4 P56524 8/20 0.38
HDAC6 Q9UBN7 8/20 0.38
HDAC3 O15379 8/20 0.38
HDAC2 Q92769 7/20 0.38
HDAC7 Q8WUI4 6/20 0.38
HDAC10 Q969S8 6/20 0.38
HDAC11 Q96DB2 6/20 0.38
HDAC8 Q9BY41 6/20 0.38
HDAC9 Q9UKV0 6/20 0.38
HDAC5 Q9UQL6 6/20 0.38
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2098051 1.00 PIN1 (0.42) PIN1HDAC1HDAC4HDAC6HDAC3
SCHEMBL2054846 0.92 HDAC1 (0.43) HDAC1HDAC4HDAC6HDAC3HDAC2
SCHEMBL2097013 0.89 HDAC1 (0.41) HDAC1HDAC4HDAC6HDAC3HDAC2
SCHEMBL2097015 0.89 HDAC1 (0.41) HDAC1HDAC4HDAC6HDAC3HDAC2
SCHEMBL2098055 0.87 PIN1 (0.42) PIN1HDAC1HDAC4HDAC6HDAC3
SCHEMBL2101048 0.84 PIN1 (0.44) PIN1HDAC1HDAC4HDAC6HDAC3
SCHEMBL2101045 0.84 PIN1 (0.44) PIN1HDAC1HDAC4HDAC6HDAC3
SCHEMBL2098056 0.81 PIN1 (0.41) PIN1HDAC1HDAC4
SCHEMBL2097882 0.81 PIN1 (0.54) PIN1HDAC1HDAC4HDAC6HDAC3
SCHEMBL14383615 0.78 PIN1 (0.49) PIN1HDAC1HDAC4HDAC6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730298-B1 SPECIFIC SUBSTRATES FOR O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE EPFL ECOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (CH) 2015-11-11 EP disclosed
US-8163479-B2 Specific substrates for O6-alkylguanine-DNA alkyltransferase ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2012-04-24 US disclosed
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase EPFL ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2007-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase AGT, AGXT, AGTR1 PIN1 2756/4885HDAC1 3223/4885HDAC4 4541/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.