SCHEMBL20995233

SCHEMBL20995233

CC(C)N1CCN(c2ccc(Br)c(F)c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.51
PKM P14618 1/20 0.51
KHK P50053 1/20 0.42
ALK Q9UM73 2/20 0.39
HDAC4 P56524 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
ACVR1 Q04771 4/20 0.38
TGFBR1 P36897 3/20 0.38
BMPR1B O00238 2/20 0.38
BMPR1A P36894 2/20 0.38
ACVRL1 P37023 2/20 0.38
ESRRB O95718 3/20 0.38
ESRRG P62508 3/20 0.38
KCNH2 Q12809 2/20 0.37
ACVR1B P36896 1/20 0.36
TNIK Q9UKE5 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29374099 1.00 KDM4E (0.51) KDM4EALDH1A1MAPTPKMKHK
SCHEMBL19358312 0.81 HTR3A (0.50) KDM4EALDH1A1MAPT
SCHEMBL29478226 0.81 HTR3A (0.50) KDM4EALDH1A1MAPT
SCHEMBL22171249 0.81 MAPT (0.51) KDM4EALDH1A1MAPTPKMKHK
Hydrochloric Acid SCHEMBL22165259 0.79 MAPT (0.50) KDM4EALDH1A1MAPTPKMKHK
SCHEMBL21361441 0.78 MAPT (0.49) KDM4EALDH1A1MAPTPKMALK
SCHEMBL29937495 0.78 ALDH1A1 (0.46) KDM4EALDH1A1MAPTPKM
SCHEMBL28867024 0.78 ALDH1A1 (0.46) KDM4EALDH1A1MAPTPKM
SCHEMBL28767962 0.76 KDM1A (0.36) ALDH1A1MAPTKCNH2
SCHEMBL27195824 0.76 KDM4E (0.50) KDM4EALDH1A1MAPTPKMKHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116869-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS NOVARTIS AG (CH) 2026-04-30 US disclosed
US-12466808-B2 Aminopyridine derivatives and their use as selective ALK-2 inhibitors NOVARTIS AG (CH) 2025-11-11 US disclosed
EP-4442317-A2 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS Novartis AG (CH) 2024-10-09 EP disclosed
EP-3971177-B1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS NOVARTIS AG (CH) 2024-06-26 EP disclosed
EP-3971177-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS Novartis AG (CH) 2022-03-23 EP disclosed
CN-114014844-A Aminopyridine derivatives and their use as selective ALK-2 inhibitors 诺华股份有限公司 2022-02-08 CN disclosed
CN-109641871-B Aminopyridine derivatives and their use as selective ALK-2 inhibitors 诺华股份有限公司 2021-10-22 CN disclosed
EP-3487851-B1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS NOVARTIS AG (CH) 2021-10-20 EP disclosed
US-20210155606-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS NOVARTIS AG (CH) 2021-05-27 US disclosed
US-10947218-B2 Aminopyridine derivatives and their use as selective ALK-2 inhibitors NOVARTIS AG (CH) 2021-03-16 US disclosed
US-20200299265-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS CHINA NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH CO., LTD (CN) 2020-09-24 US disclosed
US-10710980-B2 Aminopyridine derivatives and their use as selective ALK-2 inhibitors NOVARTIS AG (US) 2020-07-14 US disclosed
US-20190161474-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS CHINA NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH CO., LTD (CN) 2019-05-30 US disclosed
CN-109641871-A AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS 诺华股份有限公司 2019-04-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10710980-B2 Aminopyridine derivatives and their use as selective ALK-2 inhibitors ALK, ACVR2B, ACVR1B KDM4E 449/4885ALDH1A1 632/4885MAPT 2662/4885
US-12466808-B2 Aminopyridine derivatives and their use as selective ALK-2 inhibitors ALK, ACVR1, ACVR1B KDM4E 347/4885ALDH1A1 589/4885MAPT 2439/4885
US-10947218-B2 Aminopyridine derivatives and their use as selective ALK-2 inhibitors ALK, ACVR2B, ACVR1B KDM4E 372/4885ALDH1A1 799/4885MAPT 2337/4885
US-20200299265-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS ALK, ACVR2B, ACVR1B KDM4E 372/4885ALDH1A1 799/4885MAPT 2337/4885
US-20190161474-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS ALK, ACVR2B, ACVR1B KDM4E 449/4885ALDH1A1 632/4885MAPT 2662/4885
US-20260116869-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS ALK, ACVR1, ACVR1B KDM4E 1080/4885ALDH1A1 561/4885MAPT 4635/4885
US-20210155606-A1 AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS ALK, ACVR1, ACVR1B KDM4E 347/4885ALDH1A1 589/4885MAPT 2439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.