SCHEMBL21028015

SCHEMBL21028015

O=C(O)C1CCCc2c(Cc3cccnc3Sc3ccccc3)c3ccccc3n21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
ATM Q13315 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
KMT2A Q03164 3/20 0.34
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 2/20 0.34
GLA P06280 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
TSPO P30536 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21028018 0.86 PTGDR2 (0.34) SMN1; SMN2KMT2AMEN1LMNAMAPT
SCHEMBL21027972 0.81 PTGDR2 (0.45) KMT2AMEN1L3MBTL1RAB9APTGDR2
SCHEMBL21027857 0.77 PTGDR2 (0.47) ALDH1A1SMN1; SMN2KDM4ELMNAMAPT
SCHEMBL21027976 0.77 PTGDR2 (0.49) ATMPTGDR2CYP3A4
SCHEMBL21028291 0.74 PTGDR2 (0.42) ALDH1A1PTGDR2
SCHEMBL21028085 0.71 PTGDR2 (0.43) PTGDR2CYP3A4
SCHEMBL21027858 0.71 PTGDR2 (0.50) PTGDR2
SCHEMBL21027975 0.70 PTGDR2 (0.44) KMT2AKDM4EMEN1GLACASP1
SCHEMBL21028077 0.68 MEN1 (0.41) ALDH1A1ATMKMT2AKDM4EMEN1
SCHEMBL21028014 0.67 PTGDR2 (0.42) KMT2AMEN1RAB9APTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489235-A1 TRICYCLIC COMPOUND AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed