SCHEMBL21032563

SCHEMBL21032563

CCCCOC(=O)Cn1c(C)c(Cc2ccc3c(c2)CCS3)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 7/20 0.53
PLA2G2A P14555 2/20 0.39
ALDH1A1 P00352 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP3A4 P08684 1/20 0.36
ABCC1 P33527 1/20 0.36
PLA2G4A P47712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21032217 0.74 PTGDR2 (0.66) PTGDR2
SCHEMBL21032466 0.72 PTGDR2 (0.67) PTGDR2
SCHEMBL21032709 0.72 PTGDR2 (0.67) PTGDR2
SCHEMBL21032164 0.71 PTGDR2 (0.65) PTGDR2ALDH1A1
SCHEMBL21031858 0.70 PTGDR2 (0.51) PTGDR2
SCHEMBL21266666 0.69 PTGDR2 (1.00) PTGDR2PLA2G2A
SCHEMBL14979223 0.69 TDP1 (0.53) PTGDR2PLA2G2AALDH1A1TDP1MEN1
SCHEMBL21032568 0.69 PTGDR2 (0.38) PTGDR2MEN1KMT2A
SCHEMBL21031848 0.67 PTGDR2 (0.48) PTGDR2
SCHEMBL21031903 0.67 PTGDR2 (0.57) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489233-B1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2022-01-12 EP disclosed
EP-3489233-A1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed