SCHEMBL21032568

SCHEMBL21032568

Cc1c(Cc2ccc3c(c2)CCS3)c2cc(NC(=O)C3CC3)ccc2n1CC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 8/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPN6 P29350 1/20 0.34
LMNA P02545 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 2/20 0.33
TP53 P04637 2/20 0.33
F2 P00734 1/20 0.33
ELANE P08246 1/20 0.33
CTRB1 P17538 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
HTT P42858 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21031848 0.89 PTGDR2 (0.48) PTGDR2
SCHEMBL21031858 0.79 PTGDR2 (0.51) PTGDR2
SCHEMBL21032217 0.73 PTGDR2 (0.66) PTGDR2
SCHEMBL21031846 0.72 PTGDR2 (0.72) PTGDR2
SCHEMBL21032466 0.72 PTGDR2 (0.67) PTGDR2
SCHEMBL21032709 0.72 PTGDR2 (0.67) PTGDR2
SCHEMBL21032164 0.70 PTGDR2 (0.65) PTGDR2
SCHEMBL21032563 0.69 PTGDR2 (0.53) PTGDR2MEN1KMT2A
SCHEMBL21031903 0.67 PTGDR2 (0.57) PTGDR2
SCHEMBL21032593 0.66 PTGDR2 (0.48) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489233-B1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2022-01-12 EP disclosed
EP-3489233-A1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed