SCHEMBL21034080

SCHEMBL21034080

COc1ccccc1C(C)(C)C(=O)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 3/20 0.46
GAA P10253 4/20 0.44
CA12 O43570 3/20 0.44
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA9 Q16790 3/20 0.44
CA7 P43166 2/20 0.44
CA14 Q9ULX7 2/20 0.44
POLB P06746 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 2/20 0.42
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CA4 P22748 1/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 3/20 0.41
ATM Q13315 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17102000 0.85 KMT2A (0.49) KMT2AMEN1ALDH1A1GAACA12
SCHEMBL12260657 0.81 ATM (0.46) KMT2AMEN1ALDH1A1GAACA12
SCHEMBL27471238 0.80 GAA (0.49) KMT2AMEN1ALDH1A1GAACA12
SCHEMBL18493202 0.80 KMT2A (0.50) KMT2AMEN1ALDH1A1GAACA12
SCHEMBL21034079 0.79 MEN1 (0.51) KMT2AMEN1ALDH1A1GAAPOLB
SCHEMBL6404528 0.76 KMT2A (0.51) KMT2AMEN1ALDH1A1GAACA12
SCHEMBL420634 0.76 KMT2A (0.51) KMT2AMEN1ALDH1A1GAACA12
SCHEMBL11023514 0.75 KMT2A (0.47) KMT2AMEN1ALDH1A1GAACA12
SCHEMBL16672585 0.75 CNR2 (0.49) KMT2AMEN1GAAPOLBLMNA
SCHEMBL9577269 0.74 KCNN4 (0.41) KMT2AALDH1A1POLBL3MBTL1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111372936-B Mcl-1 selective inhibitors, their preparation and use 北京赛林泰医药技术有限公司 2022-12-02 CN disclosed
CN-111372936-A Mcl-1 selective inhibitors, their preparation and use 北京赛林泰医药技术有限公司 2020-07-03 CN disclosed
CN-110452253-A Mcl-1 selective depressant and its preparation and use CENTAURUS BIOPHARMA CO LTD 2019-11-15 CN disclosed
WO-2019101144-A1 SELECTIVE MCL-1 INHIBITOR AND PREPARATION AND USE THEREOF 北京赛林泰医药技术有限公司 2019-05-31 WO disclosed
CN-109824690-A Mcl-1 selective depressant and its preparation and use 北京赛林泰医药技术有限公司 2019-05-31 CN disclosed