SCHEMBL21036475

SCHEMBL21036475

CC(=O)N[C@@H](CC(C)(C)C)C(=O)N1CCNC[C@H]1C

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PLD1 Q13393 1/20 0.36
DPP4 P27487 2/20 0.35
SIGMAR1 Q99720 1/20 0.30
F2 P00734 1/20 0.30
F9 P00740 1/20 0.30
F10 P00742 1/20 0.30
F12 P00748 1/20 0.30
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
F7 P08709 1/20 0.30
PRSS3 P35030 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21124325 1.00 PLD1 (0.36) PLD1DPP4SIGMAR1F2F9
SCHEMBL18096136 0.80 DPP4 (0.38) PLD1DPP4SIGMAR1F2F9
SCHEMBL19806290 0.80 SIGMAR1 (0.30) SIGMAR1
SCHEMBL21036085 0.78 SIGMAR1 (0.37) SIGMAR1F2
SCHEMBL31591902 0.77 HDAC8 (0.42) PLD1
SCHEMBL27041826 0.75 PLD1 (0.38) PLD1DPP4
SCHEMBL20994238 0.73 CYP3A4 (0.40) PLD1
SCHEMBL21124129 0.73 PLD1 (0.39) PLD1DPP4SIGMAR1
SCHEMBL21124125 0.73 PLD1 (0.39) PLD1DPP4SIGMAR1
SCHEMBL20994235 0.73 CYP3A4 (0.40) PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489231-B1 PIPERAZINE DERIVATIVE ASTELLAS PHARMA INC (JP) 2021-06-09 EP disclosed
EP-3489231-A1 PIPERAZINE DERIVATIVE Astellas Pharma Inc. (JP) 2019-05-29 EP disclosed