SCHEMBL21044015

SCHEMBL21044015

COC(=O)C(C)(C)c1csc(NS(=O)(=O)C2CC2)n1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTPS1 P17812 18/20 0.58
CTPS2 Q9NRF8 4/20 0.58
ATAD2 Q6PL18 1/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21044406 0.95 CTPS1 (0.54) CTPS1CTPS2ATAD2MEN1KMT2A
SCHEMBL22869109 0.95 CTPS1 (0.54) CTPS1CTPS2ATAD2MEN1KMT2A
SCHEMBL21044432 0.87 CTPS1 (0.58) CTPS1CTPS2ATAD2MEN1KMT2A
SCHEMBL21044107 0.86 CTPS1 (0.58) CTPS1CTPS2ATAD2
SCHEMBL22869127 0.83 KMT2A (0.43) CTPS1CTPS2ATAD2MEN1KMT2A
SCHEMBL22490762 0.83 CTPS1 (0.53) CTPS1CTPS2ATAD2MEN1KMT2A
SCHEMBL21044343 0.82 CTPS1 (0.53) CTPS1CTPS2ATAD2
SCHEMBL22869143 0.82 CTPS1 (0.53) CTPS1CTPS2ATAD2
SCHEMBL21044009 0.82 CTPS1 (0.44) CTPS1CTPS2ATAD2MEN1KMT2A
SCHEMBL22490834 0.81 CTPS1 (0.51) CTPS1CTPS2ATAD2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3717459-B1 COMPOUNDS STEP PHARMA S A S (FR) 2026-01-21 EP disclosed
US-12503466-B2 Aminothiazole compounds as inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2025-12-23 US disclosed
US-20240010645-A1 Aminothiazole Compounds as Inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2024-01-11 US disclosed
US-11655246-B2 Aminothiazole compounds as inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2023-05-23 US disclosed
US-11655246-B2 Aminothiazole compounds as inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2023-05-23 US disclosed
US-11655246-B2 Aminothiazole compounds as inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2023-05-23 US disclosed
US-20210002269-A1 COMPOUNDS STEP PHARMA S.A.S. (FR) 2021-01-07 US disclosed
US-20210002269-A1 COMPOUNDS STEP PHARMA S.A.S. (FR) 2021-01-07 US disclosed
EP-3717459-A1 COMPOUNDS Step Pharma S.A.S. (FR) 2020-10-07 EP disclosed
EP-3492454-A1 COMPOUNDS Step Pharma S.A.S. (FR) 2019-06-05 EP disclosed
EP-3492454-A1 COMPOUNDS Step Pharma S.A.S. (FR) 2019-06-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12503466-B2 Aminothiazole compounds as inhibitors of CTPS1 CTPS1, CTPS2, TBXAS1 CTPS1 1/4885CTPS2 2/4885ATAD2 986/4885
US-11655246-B2 Aminothiazole compounds as inhibitors of CTPS1 CTPS1, CTPS2, TBXAS1 CTPS1 1/4885CTPS2 2/4885ATAD2 986/4885
US-20210002269-A1 COMPOUNDS UGT1A1, CYP1A1, CYP19A1 CTPS1 2385/4885CTPS2 2441/4885ATAD2 3919/4885
US-20240010645-A1 Aminothiazole Compounds as Inhibitors of CTPS1 CTPS1, CTPS2, TBXAS1 CTPS1 1/4885CTPS2 2/4885ATAD2 986/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.