SCHEMBL21044565

SCHEMBL21044565

COC(=O)c1cc(-n2cc(-c3ccccc3)nn2)cc(C(=O)OC)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OGT O15294 3/20 0.53
PTGS2 P35354 2/20 0.49
PTGS1 P23219 1/20 0.49
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP1B1 Q16678 1/20 0.48
STIM1 Q13586 4/20 0.47
ORAI1 Q96D31 4/20 0.47
CA12 O43570 2/20 0.46
CA2 P00918 2/20 0.46
CA9 Q16790 2/20 0.46
CA1 P00915 1/20 0.46
CA5A P35218 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
ABCB1 P08183 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
NOTUM Q6P988 2/20 0.45
HDAC3 O15379 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19182235 0.85 OGT (0.52) OGTPTGS2PTGS1CA12CA2
SCHEMBL1694849 0.82 OGT (0.48) OGTPTGS2PTGS1ALDH1A1KDM4E
SCHEMBL10120527 0.82 ABCG2 (0.46) OGTALDH1A1KDM4EHPGDHSD17B10
SCHEMBL17071962 0.79 SNCA (0.40) OGTPTGS2PTGS1CYP1B1STIM1
SCHEMBL31581056 0.79 STIM1 (0.46) OGTSTIM1ORAI1CA12CA9
SCHEMBL14836638 0.79 CYP1B1 (0.57) PTGS2PTGS1CYP1B1STIM1ORAI1
SCHEMBL1694856 0.75 KDM4E (0.55) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL17069699 0.75 SNCA (0.38) OGTPTGS2PTGS1CYP1B1STIM1
SCHEMBL4265804 0.75 ALDH1A1 (0.57) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL12571591 0.75 CA12 (0.66) KDM4ECA12CA2CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191451-B1 4-SUBSTITUTED PYRIDINE-2,6-DICARBOXYLIC ACID DERIVATIVES AND METHOD OF PREPARING SAME OKINAWA INST SCIENCE & TECH SCHOOL CORP (JP) 2019-06-05 EP claimed