SCHEMBL10120527

SCHEMBL10120527

COC(=O)c1cc(-n2cc(-c3ccccc3)nn2)c2ccccc2n1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.46
ABCB1 P08183 1/20 0.46
LDHA P00338 1/20 0.46
ALDH1A1 P00352 5/20 0.44
KDM4E B2RXH2 4/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 1/20 0.44
BCHE P06276 1/20 0.43
OGT O15294 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MIF P14174 1/20 0.41
PLA2G2A P14555 1/20 0.41
ALDH1A3 P47895 1/20 0.41
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10120532 0.89 NOTUM (0.42) ABCG2KDM4EBCHEOGTMEN1
SCHEMBL1694971 0.87 LDHA (0.53) ABCG2ABCB1LDHAKDM4EBCHE
SCHEMBL21044565 0.82 OGT (0.53) ABCG2ABCB1ALDH1A1KDM4EHPGD
SCHEMBL1694856 0.80 KDM4E (0.55) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL1695207 0.76 KMO (0.51) LDHABCHEMEN1KMT2AMIF
SCHEMBL1694849 0.75 OGT (0.48) ALDH1A1KDM4EOGTMEN1KMT2A
SCHEMBL13188224 0.73 GRM2 (0.55) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4265804 0.70 ALDH1A1 (0.57) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL2467305 0.70 ALDH1A1 (0.65) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL72379 0.70 KDM4E (0.70) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006068-A2 COMPOUNDS FOR THE INHIBITION OF CELLULAR PROLIFERATION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-12 WO disclosed