SCHEMBL21048924

SCHEMBL21048924

CCS(=O)(=O)Nc1ccc(C)cc1CNC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 1/20 0.42
HSP90AA1 P07900 1/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
XBP1 P17861 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MRGPRX1 Q96LB2 2/20 0.42
KDM4A O75164 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
HPGD P15428 2/20 0.37
EPHX2 P34913 1/20 0.37
NR1H4 Q96RI1 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21048803 0.92 TP53 (0.40) HSD17B10LMNATP53HSP90AA1GAA
SCHEMBL17258751 0.84 KCNA5 (0.46) LMNAKDM4AHPGDKDM4EALDH1A1
SCHEMBL5015072 0.80 NPC1 (0.54) HSD17B10LMNATP53HSP90AA1GAA
SCHEMBL31705342 0.77 KDM4A (0.44) GAAKDM4AALDH1A1NQO2KCNA5
SCHEMBL13104124 0.77 KDM4A (0.44) GAAKDM4AKCNA5NPC1RAB9A
SCHEMBL15171404 0.76 NPC1 (0.52) KDM4ASMN1; SMN2EPHX2KDM4EALDH1A1
SCHEMBL21048807 0.76 KCNA5 (0.43) LMNAKDM4AHPGDKDM4EALDH1A1
SCHEMBL27669339 0.76 KDM4A (0.43) HSD17B10LMNATP53HSP90AA1GAA
SCHEMBL21048804 0.75 JAK2 (0.41) HSD17B10LMNATP53HSP90AA1GAA
SCHEMBL21048954 0.75 LMNA (0.38) HSD17B10LMNATP53HSP90AA1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143021-B1 PYRAZOLOPYRIDINES AND PYRAZOLOPYRIMIDINES PFIZER (US) 2019-06-12 EP disclosed