SCHEMBL210527

SCHEMBL210527

O=C(CN1CCN(C(=O)O)CC1)Nc1nccs1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 8/20 0.64
LMNA P02545 2/20 0.60
KMT2A Q03164 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.58
KDR P35968 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15134850 0.86 KCNA5 (0.69) KCNA5LMNAKMT2ASMN1; SMN2
SCHEMBL10282572 0.85 KCNA5 (0.64) KCNA5LMNAKMT2ASMN1; SMN2
SCHEMBL27635088 0.83 KCNA5 (0.60) KCNA5LMNAKMT2ASMN1; SMN2
SCHEMBL654947 0.82 KCNA5 (0.59) KCNA5LMNAKMT2ASMN1; SMN2
SCHEMBL14520853 0.82 KCNA5 (0.53) KCNA5LMNAKMT2ASMN1; SMN2
SCHEMBL210449 0.82 KCNA5 (0.59) KCNA5LMNAKMT2A
SCHEMBL5329430 0.82 KCNA5 (0.53) KCNA5LMNAKMT2ASMN1; SMN2
SCHEMBL10245284 0.82 KCNA5 (0.62) KCNA5LMNAKMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL207813 0.81 KCNA5 (0.58) KCNA5LMNAKMT2ASMN1; SMN2
SCHEMBL10282859 0.81 LMNA (0.62) KCNA5LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963315-B1 ENZYME INHIBITORS CANCER REC TECH LTD (GB) 2014-10-08 EP disclosed
US-8088761-B2 Enzyme inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2012-01-03 US disclosed
US-20090247507-A1 Enzyme Inhibitors THE INSTITUTE OF CANCER RESEARCH (GB) 2009-10-01 US disclosed
EP-1963315-A2 ENZYME INHIBITORS The Institute of Cancer Research (GB) 2008-09-03 EP disclosed
WO-2007072017-A2 ENZYME INHIBITORS THE INSTITUTE OF CANCER RESEARCH (GB) 2007-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090247507-A1 Enzyme Inhibitors AURKC, AURKB, AURKA KCNA5 1499/4885LMNA 2674/4885KMT2A 384/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.