Azaconazole

Azaconazole

SCHEMBL2364039

Clc1ccc(C2(Cn3cncn3)OCCO2)c(Cl)c1.c1c[nH]nn1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 15/20 0.56
THRB P10828 1/20 0.56
CYP2C9 P11712 2/20 0.50
LMNA P02545 2/20 0.44
FYN P06241 2/20 0.44
CYP51A1 Q16850 2/20 0.44
NR1I2 O75469 1/20 0.44
PGR P06401 1/20 0.44
HSP90AA1 P07900 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
ADRA2A P08913 1/20 0.44
CHRM1 P11229 1/20 0.44
TSHR P16473 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
CHRM3 P20309 1/20 0.44
DRD1 P21728 1/20 0.44
TBXA2R P21731 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Azaconazole SCHEMBL21056 0.88 CYP3A4 (0.69) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL3009257 0.88 CYP3A4 (0.69) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL29354903 0.88 CYP3A4 (0.69) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL29017725 0.87 CYP3A4 (0.67) CYP3A4THRBCYP2C9LMNAFYN
Etaconazole SCHEMBL10335839 0.85 CYP3A4 (0.81) CYP3A4THRBCYP2C9LMNAFYN
SCHEMBL2127240 0.84 CYP3A4 (0.66) CYP3A4THRBCYP2C9LMNAFYN
Propiconazole SCHEMBL693848 0.83 CYP3A4 (0.82) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL11544952 0.82 CYP3A4 (0.61) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL11543267 0.81 KDM4E (0.60) CYP3A4THRBCYP2C9LMNAFYN
SCHEMBL11540746 0.79 CYP3A4 (0.56) CYP3A4THRBCYP2C9LMNAFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072634-A2 POST-HARVEST TREATMENT METHOD BASF SE (DE) 2010-07-01 WO claimed
WO-2011094219-A1 VESICULAR FORMULATIONS KROON HENDRICK-ANDRE (US) 2011-08-04 WO disclosed