SCHEMBL21064707

SCHEMBL21064707

Cc1cn(C(C)C(=O)N(C)C)cn1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 2/20 0.33
CCNC P24863 3/20 0.32
CDK8 P49336 3/20 0.32
ALPL P05186 2/20 0.31
PLAA Q9Y263 1/20 0.31
SYK P43405 1/20 0.30
ALPG P10696 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20008981 0.85 CPA1 (0.34) KDM5ACCNCCDK8
SCHEMBL4453713 0.80 ALDH1A1 (0.41) KDM5AALPLPLAAALPGALDH1A1
SCHEMBL20012745 0.79 KDM5A (0.31) KDM5ACCNCCDK8
SCHEMBL1507952 0.71 FAAH (0.36) ALPLPLAAALPGALDH1A1
SCHEMBL18038750 0.69
SCHEMBL14857100 0.68 KDM5A (0.32) KDM5AALPLPLAAALPGALDH1A1
SCHEMBL14857102 0.68 KDM5A (0.32) KDM5AALPLPLAAALPGALDH1A1
SCHEMBL26186634 0.68 CYP2E1 (0.30)
SCHEMBL21149908 0.67
SCHEMBL20306252 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3262036-B1 THERAPEUTIC PYRIDAZINE COMPOUNDS AND USES THEREOF GENENTECH INC (US) 2023-09-13 EP disclosed
US-10308614-B2 Therapeutic compounds and uses thereof GENENTECH, INC. (US) 2019-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10308614-B2 Therapeutic compounds and uses thereof SMARCC1, SMARCC2, SMARCA4 KDM5A 1915/4885CCNC 3381/4885CDK8 1604/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.