SCHEMBL21065259

SCHEMBL21065259

Cc1nc2c3ccccc3n3c4ccccc4nc3n2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 8/20 0.50
KDM4E B2RXH2 6/20 0.50
HSD17B10 Q99714 5/20 0.50
ALDH1A1 P00352 4/20 0.50
LMNA P02545 3/20 0.50
MAPT P10636 3/20 0.50
POLB P06746 3/20 0.50
TSHR P16473 2/20 0.50
TP53 P04637 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.44
HAVCR2 Q8TDQ0 1/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
PDE5A O76074 1/20 0.39
PDE1B Q01064 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL861183 0.76 KDM4E (0.57) KDM4EHSD17B10ALDH1A1LMNAMAPT
SCHEMBL21065258 0.75 KMT2A (0.58) KDM4EHSD17B10ALDH1A1LMNAMAPT
SCHEMBL12759656 0.73 HSD17B10 (0.56) PDE10AKDM4EHSD17B10ALDH1A1LMNA
SCHEMBL24848571 0.72 KDM4E (0.49) KDM4EHSD17B10ALDH1A1LMNAMAPT
SCHEMBL17993463 0.71 KDM4E (0.65) KDM4EHSD17B10ALDH1A1LMNAMAPT
SCHEMBL18057364 0.71 KDM4E (0.60) KDM4EHSD17B10ALDH1A1LMNAMAPT
SCHEMBL12838246 0.71 PDE10A (0.67) PDE10AKDM4EHSD17B10LMNAMAPT
SCHEMBL24848558 0.70 KDM4E (0.46) PDE10AKDM4EHSD17B10ALDH1A1LMNA
SCHEMBL11169562 0.70 HSD17B10 (0.52) PDE10AKDM4EHSD17B10ALDH1A1LMNA
SCHEMBL7398110 0.69 PDE10A (0.63) PDE10AKDM4EHSD17B10LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399922-B1 Metal complexes of cyclometallated imidazo(1,2-f) phenanthridine and diimidazo(1,2-A;1',2'-C)quinazoline ligands and isoelectronic and benzannulated analogs therof UNIVERSAL DISPLAY CORP (US) 2019-06-26 EP claimed
EP-2399922-B1 Metal complexes of cyclometallated imidazo(1,2-f) phenanthridine and diimidazo(1,2-A;1',2'-C)quinazoline ligands and isoelectronic and benzannulated analogs therof UNIVERSAL DISPLAY CORP (US) 2019-06-26 EP disclosed