SCHEMBL21074459

SCHEMBL21074459

C/N=C(\C)c1cc(C)cc(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.39
GAA P10253 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
RAPGEF4 Q8WZA2 1/20 0.36
GRIN2B Q13224 1/20 0.36
ADCY8 P40145 2/20 0.35
ADCY1 Q08828 2/20 0.35
PGK1 P00558 1/20 0.35
PGK2 P07205 1/20 0.35
KCNK3 O14649 1/20 0.34
KCNK9 Q9NPC2 1/20 0.34
HTT P42858 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
NOTUM Q6P988 2/20 0.33
TAS2R14 Q9NYV8 1/20 0.33
AKT1 P31749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12288118 0.88 CES2 (0.50) CES2GAAMEN1KMT2ACTSL
SCHEMBL2365619 0.88 CES2 (0.50) CES2GAAMEN1KMT2ACTSL
SCHEMBL17191009 0.85 SMN1; SMN2 (0.42) CES2GAAMEN1KMT2ACTSL
SCHEMBL16962044 0.80 CES2 (0.45) CES2CTSLCTSBRAPGEF4GRIN2B
SCHEMBL13954751 0.77 CES2 (0.42) CES2CTSLCTSBRAPGEF4GRIN2B
SCHEMBL17586584 0.77 CES2 (0.57) CES2GAARAPGEF4ADCY8ADCY1
SCHEMBL7786247 0.77 CES2 (0.52) CES2MEN1KMT2AADCY8ADCY1
SCHEMBL23526049 0.76 CES2 (0.33) CES2GAAMEN1KMT2ACTSL
SCHEMBL23526051 0.76 CES2 (0.33) CES2GAAMEN1KMT2ACTSL
SCHEMBL23526054 0.76 CES2 (0.33) CES2GAAMEN1KMT2ACTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3492455-A1 1,2,4-TRIAZOLES AS NUCLEAR TRANSPORT MODULATORS AND USE IN THE TREATMENT OF SPECIFIC FORMS OF CANCER Karyopharm Therapeutics Inc. (US) 2019-06-05 EP disclosed