SCHEMBL21077925

SCHEMBL21077925

N#CC1(c2ccccc2)CCN(I)CC1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.61
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA9 Q16790 1/20 0.58
OPRD1 P41143 1/20 0.55
OPRL1 P41146 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL56575 0.82 NPC1 (0.57) OPRM1CA12CA1CA2CA9
SCHEMBL872608 0.82 OPRM1 (0.56) OPRM1CA12CA1CA2CA9
SCHEMBL432561 0.82 OPRM1 (0.59) OPRM1CA12CA1CA2CA9
SCHEMBL504355 0.81 OPRM1 (0.70) OPRM1CA12CA1CA2CA9
SCHEMBL11211164 0.81 OPRM1 (0.61) OPRM1CA12CA1CA2CA9
SCHEMBL13548727 0.81 OPRM1 (0.66) OPRM1CA12CA1CA2CA9
SCHEMBL18768887 0.80 NPC1 (0.55) OPRM1CA12CA1CA2CA9
SCHEMBL19249603 0.80 NPC1 (0.55) OPRM1CA12CA1CA2CA9
SCHEMBL181145 0.80 NPC1 (0.55) OPRM1CA12CA1CA2CA9
SCHEMBL8580359 0.80 CA12 (0.60) OPRM1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3145929-B1 5-CHLORO-2-DIFLUOROMETHOXYPHENYL PYRAZOLOPYRIMIDINE COMPOUNDS WHICH ARE JAK INHIBITORS HOFFMANN LA ROCHE (CH) 2021-01-13 EP disclosed
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed