SCHEMBL21077978

SCHEMBL21077978

CSc1ccc(C(=O)C2CCCC3(CC2)CNC3)cc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 3/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
LMNA P02545 2/20 0.42
SLC18A3 Q16572 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 5/20 0.40
MEN1 O00255 3/20 0.40
CYP2D6 P10635 1/20 0.40
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5187550 0.80 ALDH1A1 (0.57) ALDH1A1KDM4EPOLBRXFP1MAPT
SCHEMBL6988277 0.80 ALDH1A1 (0.57) ALDH1A1KDM4EPOLBRXFP1MAPT
SCHEMBL2993708 0.79 SRD5A2 (0.57) ALDH1A1KDM4EPOLBRXFP1MAPT
SCHEMBL5187629 0.77 SLC18A3 (0.56) ALDH1A1KDM4EPOLBRXFP1LMNA
SCHEMBL13874024 0.76 MEN1 (0.66) ALDH1A1KDM4EPOLBRXFP1MAPT
Hydrochloric Acid SCHEMBL3846012 0.75 MEN1 (0.69) ALDH1A1KDM4EPOLBRXFP1MAPT
SCHEMBL4771785 0.67 SLC18A3 (0.56) ALDH1A1KDM4EPOLBRXFP1SLC18A3
SCHEMBL2989814 0.65 PLK1 (0.44) ALDH1A1KDM4EPOLBRXFP1MAPT
SCHEMBL21078129 0.65 SLC18A3 (0.45) ALDH1A1KDM4EPOLBRXFP1MAPT
SCHEMBL29967623 0.63 KMT2A (0.41) KDM4EMAPTLMNASMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed