SCHEMBL21083380

SCHEMBL21083380

Cc1ccc2ncc(C(=O)NCCN3CCOCC3)n2c1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.66
RAB9A P51151 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
PIK3CD O00329 1/20 0.52
PIK3R1 P27986 1/20 0.52
PIK3CA P42336 1/20 0.52
PIK3CB P42338 1/20 0.52
PIK3CG P48736 1/20 0.52
ALDH1A1 P00352 1/20 0.52
POLB P06746 2/20 0.51
TSHR P16473 1/20 0.49
KDM5B Q9UGL1 1/20 0.48
CD274 Q9NZQ7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21084195 0.87 TGFBR1 (0.61) TGFBR1PIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL22955513 0.86 TGFBR1 (0.60) TGFBR1PIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL24654175 0.86 TGFBR1 (0.60) TGFBR1PIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL21084232 0.80 TGFBR1 (1.00) TGFBR1
SCHEMBL16917273 0.80 TGFBR1 (0.62) TGFBR1PIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL22955994 0.80 TGFBR1 (1.00) TGFBR1PIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL22955787 0.80 TGFBR1 (0.67) TGFBR1PIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL21084064 0.77 TGFBR1 (0.63) TGFBR1ALDH1A1
SCHEMBL30117458 0.76 TGFBR1 (0.64) TGFBR1PIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL15638831 0.76 TGFBR1 (0.64) TGFBR1PIK3CDPIK3R1PIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3492461-A1 NITROGENOUS HETEROCYCLIC AROMATIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF Shanghai Yingli Pharmaceutical Co. Ltd. (CN) 2019-06-05 EP disclosed