Xanoxic Acid

Xanoxic Acid

SCHEMBL2109668

CC(C)Oc1ccc2oc3ccc(C(=O)O)cc3c(=O)c2c1

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.88
KDM4E B2RXH2 3/20 0.88
HPGD P15428 3/20 0.88
KMT2A Q03164 2/20 0.88
MEN1 O00255 1/20 0.88
TP53 P04637 1/20 0.88
CYP2C9 P11712 1/20 0.88
PTGER1 P34995 1/20 0.88
PTGER3 P43115 1/20 0.88
PTGER2 P43116 1/20 0.88
PTGDR Q13258 1/20 0.88
HSD17B10 Q99714 1/20 0.88
TTR P02766 7/20 0.61
AKR1B1 P15121 1/20 0.54
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
MAPT P10636 1/20 0.53
CASP3 P42574 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
SENP8 Q96LD8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1163801 0.93 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL29627447 0.93 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL10453911 0.93 KDM4E (0.90) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL10454176 0.92 KDM4E (0.88) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL10454177 0.92 KDM4E (0.88) ALDH1A1KDM4EHPGDKMT2AMEN1
Xanoxic Acid SCHEMBL29400285 0.86 ALDH1A1 (0.67) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL11768660 0.86 ALDH1A1 (0.67) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL11768887 0.86 KMT2A (0.67) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL10785566 0.86 ALDH1A1 (0.66) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL1105126 0.86 KDM4E (0.73) ALDH1A1KDM4EHPGDKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
CN-102149282-A Carbonate prodrugs and methods of using the same NEUROGESX INC 2011-08-10 CN claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
EP-0028410-B1 USE OF THROMBOXANE-SYNTHETASE INHIBITING COMPOUNDS IN THE TREATMENT OF OBESITY AND THE LOWERING OF INSULIN LEVELS F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1987-09-30 EP claimed
EP-0028410-A1 Use of thromboxane-synthetase inhibiting compounds in the treatment of obesity and the lowering of insulin levels F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-05-13 EP claimed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 US disclosed
US-11191719-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2021-12-07 US disclosed
US-10463611-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2019-11-05 US disclosed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US disclosed
CN-102149282-B Carbonate prodrugs and methods of using the same NEUROGESX INC 2014-12-17 CN disclosed
US-4626432-A 7-HYDROXY-OR ALKOXYXANTHONE-2-CARBOXYLIC ACID BURROUGHS WELLCOME CO. (US) 1986-12-02 US disclosed
US-4591594-A INSULIN LOWERING AGENTS HOFFMANN-LA ROCHE INC. (US) 1986-05-27 US disclosed
US-4500540-A DIETETICS HOFFMANN-LA ROCHE INC. (US) 1985-02-19 US disclosed
EP-0028410-A1 Use of thromboxane-synthetase inhibiting compounds in the treatment of obesity and the lowering of insulin levels F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-05-13 EP disclosed
EP-0028410-A1 Use of thromboxane-synthetase inhibiting compounds in the treatment of obesity and the lowering of insulin levels F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-05-13 EP disclosed