SCHEMBL21098792

SCHEMBL21098792

CCCC(=O)N(C=O)OC(=O)CCCOc1ccc2c(c1)CCCCC2=N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.41
SLC2A1 P11166 1/20 0.36
MAOB P27338 4/20 0.35
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
PPARD Q03181 4/20 0.34
MAOA P21397 1/20 0.34
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
PDK2 Q15119 1/20 0.34
PPARA Q07869 2/20 0.33
PPARG P37231 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21099229 0.77 KMT2A (0.41) BRD4KDM4EPOLBMEN1NPC1
SCHEMBL21098772 0.76 BRD4 (0.39) BRD4SLC2A1PDK2MEN1NPC1
SCHEMBL21098795 0.75 MAOB (0.44) MAOBHRH3PPARDMAOAPPARG
SCHEMBL21098941 0.74 MAOA (0.49) MAOBKDM4EPOLBPPARDMAOA
SCHEMBL21052076 0.71 BRD4 (0.71) BRD4MAOBHRH3MAOAPDE3B
SCHEMBL22815609 0.66 BRD4 (0.82) BRD4MAOBHRH3MAOAPDE3B
SCHEMBL20010711 0.65 CYP1A2 (0.49) THRBALDH1A1MAPTKMT2A
SCHEMBL21098679 0.64 MAOB (0.63) MAOBHRH3MAOA
SCHEMBL24101995 0.64 CYP1A2 (0.43) THRBMEN1ALDH1A1MAPTKMT2A
SCHEMBL18458260 0.63 KMT2A (0.39) GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019109188-A1 ACYL HYDRAZONE LINKERS, METHODS AND USES THEREOF ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR) (CA) 2019-06-13 WO disclosed