SCHEMBL21100366

SCHEMBL21100366

C=C(NCCCc1ccc(-c2ccccc2F)cc1)C1CCN(C)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.41
GRIA4 P48058 1/20 0.40
ASAH1 Q13510 5/20 0.40
KDM1A O60341 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
MAPKAPK2 P49137 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
WNT1 P04628 1/20 0.39
DYRK1A Q13627 1/20 0.39
GBA1 P04062 1/20 0.39
UGCG Q16739 1/20 0.39
GBA2 Q9HCG7 1/20 0.39
DAO P14920 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29411602 0.87 ALDH1A1 (0.48) HTR3AKDM1AMAOAMAOBMEN1
SCHEMBL21045499 0.87 ALDH1A1 (0.48) HTR3AKDM1AMAOAMAOBMEN1
SCHEMBL21045324 0.72 NAMPT (0.48) GRIA4ASAH1MEN1ALDH1A1CYP3A4
SCHEMBL29411378 0.72 NAMPT (0.48) GRIA4ASAH1MEN1ALDH1A1CYP3A4
SCHEMBL21045114 0.71 FKBP1A (0.57) POLB
SCHEMBL21045115 0.71 FKBP1A (0.57) POLB
SCHEMBL29411452 0.71 FKBP1A (0.57) POLB
SCHEMBL21045374 0.71 ALDH1A1 (0.47) HTR3AGRIA4ASAH1MEN1ALDH1A1
SCHEMBL21045199 0.71 ALDH1A1 (0.47) HTR3AGRIA4ASAH1MEN1ALDH1A1
SCHEMBL21045200 0.71 ALDH1A1 (0.47) HTR3AGRIA4ASAH1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019113242-A1 TUBULIN INHIBITORS Lin BioScience, LLC (US) 2019-06-13 WO disclosed