SCHEMBL21101366

SCHEMBL21101366

CC(C)(C)OC(=O)N1CCC(CN(C(=O)C(F)(F)F)C2CC2)C1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
NR1H2 P55055 1/20 0.39
GPR119 Q8TDV5 5/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
USP30 Q70CQ3 2/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
HPGD P15428 1/20 0.39
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
RECQL P46063 1/20 0.37
EPHX1 P07099 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23924565 0.91 NR1H2 (0.45) JAK2JAK1NR1H2GPR119MEN1
SCHEMBL21101365 0.88 NR1H2 (0.40) NR1D1JAK2JAK1NR1H2GPR119
SCHEMBL24033522 0.82 NR1H2 (0.44) NR1D1JAK2JAK1NR1H2GPR119
SCHEMBL24033340 0.82 NR1H2 (0.44) NR1D1JAK2JAK1NR1H2GPR119
SCHEMBL21101363 0.81 USP2 (0.40) JAK2JAK1GPR119USP30MEN1
SCHEMBL1996182 0.80 NR1H2 (0.48) NR1D1JAK2JAK1NR1H2GPR119
SCHEMBL3568388 0.80 NR1H2 (0.48) NR1D1JAK2JAK1NR1H2GPR119
SCHEMBL3564630 0.80 NR1H2 (0.48) NR1D1JAK2JAK1NR1H2GPR119
SCHEMBL15411988 0.79 RORC (0.48) NR1D1JAK2JAK1GPR119KDM4E
SCHEMBL15411990 0.79 RORC (0.48) NR1D1JAK2JAK1GPR119KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2688568-B1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2019-06-19 EP disclosed