Asobamast

Asobamast

SCHEMBL2111159

CCOCCOC(=O)C(=O)Nc1nc(-c2cc(C)no2)cs1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
PKM P14618 1/20 0.44
MAPT P10636 7/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
CFTR P13569 1/20 0.41
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
PARP1 P09874 1/20 0.39
PTPN1 P18031 3/20 0.39
LMNA P02545 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPK1 P28482 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10518524 0.90 ALDH1A1 (0.59) ALDH1A1PKMMAPTNPC1RAB9A
SCHEMBL10519201 0.89 ALDH1A1 (0.44) ALDH1A1PKMMAPTNPC1RAB9A
SCHEMBL10520495 0.88 ALDH1A1 (0.43) ALDH1A1PKMMAPTNPC1RAB9A
SCHEMBL10519332 0.88 MAPT (0.45) ALDH1A1PKMMAPTNPC1RAB9A
SCHEMBL10519110 0.88 ALDH1A1 (0.42) ALDH1A1PKMMAPTNPC1RAB9A
SCHEMBL10519705 0.86 ALDH1A1 (0.41) ALDH1A1PKMMAPTNPC1RAB9A
SCHEMBL10519957 0.85 PARP1 (0.49) ALDH1A1MAPTNPC1RAB9APOLB
SCHEMBL10518463 0.82 ALDH1A1 (0.40) ALDH1A1PKMMAPTNPC1RAB9A
SCHEMBL10517375 0.82 PARP1 (0.46) ALDH1A1MAPTNPC1RAB9APOLB
SCHEMBL11141222 0.82 LMNA (0.46) ALDH1A1PKMMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2913062-B1 THERAPEUTIC OR PROPHYLACTIC AGENT FOR RETINOPATHY OF PREMATURITY AND METHOD OF TESTING FOR RETINOPATHY OF PREMATURITY JAPAN INNOVATIVE THERAPEUTICS INC (JP) 2019-05-08 EP claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 US disclosed
US-11191719-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2021-12-07 US disclosed
US-10463611-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2019-11-05 US disclosed
US-10330670-B2 Therapeutic or prophylactic agent for retinopathy of prematurity, testing method for retinopathy of prematurity, and screening method for therapeutic or prophylactic substance for retinopathy of prematurity NATIONAL UNIVERSITY CORPORATION TOKYO UNIVERSITY OF AGRICULTURE AND TECHNOLOGY (JP) 2019-06-25 US disclosed
EP-2913062-B1 THERAPEUTIC OR PROPHYLACTIC AGENT FOR RETINOPATHY OF PREMATURITY AND METHOD OF TESTING FOR RETINOPATHY OF PREMATURITY JAPAN INNOVATIVE THERAPEUTICS INC (JP) 2019-05-08 EP disclosed
US-9533056-B2 Dipeptide-based prodrug linkers for aliphatic amine-containing drugs ASCENDIS PHARMA AS (DK) 2017-01-03 US disclosed
US-4766137-A 4-(isoxazolyl)-thiazole-2-oxamic acids and derivatives thereof ZAMBON S.P.A. (IT) 1988-08-23 US disclosed
US-4766138-A Use of 4-(isoxazolyl)-thiazole-2-oxamic acid derivatives ZAMBON S.P.A. (IT) 1988-08-23 US disclosed
EP-0191045-A1 USE OF 4-(ISOXAZOLYL)-THIAZOLE-2-OXAMIC ACID DERIVATIVES. ZAMBON SPA (IT) 1986-08-20 EP disclosed
EP-0190298-A1 4-(ISOXAZOLYL)-THIAZOLE-2-OXAMIC ACIDS AND DERIVATIVES THEREOF. ZAMBON SPA (IT) 1986-08-13 EP disclosed
WO-1986000899-A1 USE OF 4-(ISOXAZOLYL)-THIAZOLE-2-OXAMIC ACID DERIVATIVES ZAMBON S.P.A. (IT) 1986-02-13 WO disclosed
WO-1986000900-A1 4-(ISOXAZOLYL)-THIAZOLE-2-OXAMIC ACIDS AND DERIVATIVES THEREOF ZAMBON, S.P.A. (IT) 1986-02-13 WO disclosed